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5CSW

B-RAF in complex with Dabrafenib

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1A, BSerine/threonine-protein kinase B-rafpolymer28232029.72UniProt (P15056)
Pfam (PF07714)
In PDB
Homo sapiens (Human)Proto-oncogene B-Raf,p94,v-Raf murine sarcoma viral oncogene homolog B1
2A, BDabrafenibnon-polymer519.62Chemie (P06)
3BCHLORIDE IONnon-polymer35.51Chemie (CL)
4waterwater18.016Chemie (HOH)
Sequence modifications
A, B: 442 - 721 (UniProt: P15056)
PDBExternal DatabaseDetails
Pro 443Arg 443engineered mutation
Ala 543Ile 543engineered mutation
Ser 544Ile 544engineered mutation
Lys 551Ile 551engineered mutation
Arg 562Gln 562engineered mutation
Asn 588Leu 588engineered mutation
Ser 630Lys 630engineered mutation
Glu 667Phe 667engineered mutation
Ser 673Tyr 673engineered mutation
Arg 688Ala 688engineered mutation
Ser 706Leu 706engineered mutation
Arg 709Gln 709engineered mutation
Glu 713Ser 713engineered mutation
Glu 716Leu 716engineered mutation
Glu 720Ser 720engineered mutation
Ser 722-expression tag
Gly 723-expression tag
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains2
Total formula weight64059.4
Non-Polymers*Number of molecules3
Total formula weight1074.6
All*Total formula weight65134.0
*Water molecules are not included.

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PDB entries from 2024-06-12

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