5AR8
RIP2 Kinase Catalytic Domain (1 - 310) complex with Biphenylsulfonamide
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | A, B | RECEPTOR-INTERACTING SERINE/THREONINE-PROTEIN KINASE 2 | polymer | 326 | 37606.0 | 2 | UniProt (O43353) Pfam (PF07714) In PDB | HOMO SAPIENS (HUMAN) | CARD-CONTAINING INTERLEUKIN-1 BETA-CONVERTING ENZYME-ASSOCI ATED KINASE, CARD-CONTAINING IL-1 BETA ICE-KINASE, RIP-LIKE-INTERA CTING CLARP KINASE, RECEPTOR-INTERACTING PROTEIN 2, RIP-2, TYROSIN E-PROTEIN KINASE RIPK2 |
2 | A, B | 2,6-bis(fluoranyl)-N-[3-[5-[2-[(3-methylsulfonylphenyl)amino]pyrimidin-4-yl]-2-morpholin-4-yl-1,3-thiazol-4-yl]phenyl]benzenesulfonamide | non-polymer | 684.8 | 2 | Chemie (XYW) | |||
3 | water | water | 18.0 | 129 | Chemie (HOH) |
Sequence modifications
A, B: 1 - 310 (UniProt: O43353)
PDB | External Database | Details |
---|---|---|
Met -15 | - | expression tag |
Asp -14 | - | expression tag |
Tyr -13 | - | expression tag |
Lys -12 | - | expression tag |
Asp -11 | - | expression tag |
Asp -10 | - | expression tag |
Asp -9 | - | expression tag |
Asp -8 | - | expression tag |
Lys -7 | - | expression tag |
Glu -6 | - | expression tag |
Asn -5 | - | expression tag |
Leu -4 | - | expression tag |
Tyr -3 | - | expression tag |
Phe -2 | - | expression tag |
Gln -1 | - | expression tag |
Gly 0 | - | expression tag |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 2 |
Total formula weight | 75212.0 | |
Non-Polymers* | Number of molecules | 2 |
Total formula weight | 1369.5 | |
All* | Total formula weight | 76581.5 |