5APK
Ligand complex of RORg LBD
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | A, B | NUCLEAR RECEPTOR ROR-GAMMA | polymer | 265 | 30918.5 | 2 | UniProt (P51449) Pfam (PF00104) In PDB | HOMO SAPIENS (HUMAN) | NUCLEAR RECEPTOR RZR-GAMMA, NUCLEAR RECEPTOR SUBFAMILY 1 GROUP F MEMBER 3, RAR-RELATED ORPHAN RECEPTOR C, RETINOID-RELATED ORPHAN RECEPTOR-GAMMA, RORG |
2 | D | NUCLEAR RECEPTOR ROR-GAMMA | polymer | 13 | 1632.9 | 1 | UniProt (P51449) In PDB | HOMO SAPIENS (HUMAN) | NUCLEAR RECEPTOR RZR-GAMMA, NUCLEAR RECEPTOR SUBFAMILY 1 GROUP F MEMBER 3, RAR-RELATED ORPHAN RECEPTOR C, RETINOID-RELATED ORPHAN RECEPTOR-GAMMA, RORG |
3 | A, B | 2-CHLORO-6-FLUORO-N-[4-[3-(TRIFLUOROMETHYL)PHENYL]SULFONYL-3,5-DIHYDRO-2H-1,4-BENZOXAZEPIN-7-YL]BENZAMIDE | non-polymer | 528.9 | 2 | Chemie (76E) | |||
4 | water | water | 18.0 | 303 | Chemie (HOH) |
Sequence modifications
A, B: 265 - 507 (UniProt: P51449)
PDB | External Database | Details |
---|---|---|
Met 243 | - | expression tag |
His 244 | - | expression tag |
Asn 245 | - | expression tag |
His 246 | - | expression tag |
Asn 247 | - | expression tag |
His 248 | - | expression tag |
Asn 249 | - | expression tag |
His 250 | - | expression tag |
Asn 251 | - | expression tag |
His 252 | - | expression tag |
Asn 253 | - | expression tag |
His 254 | - | expression tag |
Asn 255 | - | expression tag |
Gly 256 | - | expression tag |
Gly 257 | - | expression tag |
Glu 258 | - | expression tag |
Asn 259 | - | expression tag |
Leu 260 | - | expression tag |
Tyr 261 | - | expression tag |
Phe 262 | - | expression tag |
Gln 263 | - | expression tag |
Gly 264 | - | expression tag |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 3 |
Total formula weight | 63469.9 | |
Non-Polymers* | Number of molecules | 2 |
Total formula weight | 1057.8 | |
All* | Total formula weight | 64527.7 |