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4UIX

N-TERMINAL BROMODOMAIN OF HUMAN BRD4 WITH 7-(3,4-dimethoxyphenyl)-N-(1,1-dioxo-1-thian-4-yl)-5-methyl-4-oxo-4H,5H-thieno-3,2-c-pyridine-2- carboxamide

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1A, B, CBROMODOMAIN-CONTAINING PROTEIN 4polymer12715100.43UniProt (O60885)
Pfam (PF00439)
In PDB
HOMO SAPIENS (HUMAN)PROTEIN HUNK1, NHUMAN BRD4
2A, BCALCIUM IONnon-polymer40.12Chemie (CA)
3A, B, C1,2-ETHANEDIOLnon-polymer62.13Chemie (EDO)
4A, B, CN-[1,1-bis(oxidanylidene)thian-4-yl]-7-(3,4-dimethoxyphenyl)-5-methyl-4-oxidanylidene-thieno[3,2-c]pyridine-2-carboxamidenon-polymer476.63Chemie (TVU)
5waterwater18.0428Chemie (HOH)
Sequence modifications
A, B, C: 44 - 168 (UniProt: O60885)
PDBExternal DatabaseDetails
Ser 42-expression tag
Met 43-expression tag
Lys 78Gln 78conflict
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains3
Total formula weight45301.3
Non-Polymers*Number of molecules8
Total formula weight1696.1
All*Total formula weight46997.4
*Water molecules are not included.

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PDB entries from 2024-08-14

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