4N70
Pim1 Complexed with a pyridylcarboxamide
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | A | Serine/threonine-protein kinase pim-1 | polymer | 328 | 37596.7 | 1 | UniProt (P11309) Pfam (PF00069) In PDB | Homo sapiens (human) | |
2 | A | N-{4-[(3R,4R,5S)-3-amino-4-hydroxy-5-methylpiperidin-1-yl]pyridin-3-yl}-6-(2,6-difluorophenyl)-5-fluoropyridine-2-carboxamide | non-polymer | 457.4 | 1 | Chemie (2HX) | |||
3 | water | water | 18.0 | 234 | Chemie (HOH) |
Sequence modifications
A: 2 - 313 (UniProt: P11309)
PDB | External Database | Details |
---|---|---|
Met -14 | - | EXPRESSION TAG |
Ala -13 | - | EXPRESSION TAG |
His -12 | - | EXPRESSION TAG |
His -11 | - | EXPRESSION TAG |
His -10 | - | EXPRESSION TAG |
His -9 | - | EXPRESSION TAG |
His -8 | - | EXPRESSION TAG |
His -7 | - | EXPRESSION TAG |
Leu -6 | - | EXPRESSION TAG |
Glu -5 | - | EXPRESSION TAG |
Val -4 | - | EXPRESSION TAG |
Leu -3 | - | EXPRESSION TAG |
Phe -2 | - | EXPRESSION TAG |
Gln -1 | - | EXPRESSION TAG |
Gly 0 | - | EXPRESSION TAG |
Pro 1 | - | EXPRESSION TAG |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 1 |
Total formula weight | 37596.7 | |
Non-Polymers* | Number of molecules | 1 |
Total formula weight | 457.4 | |
All* | Total formula weight | 38054.2 |