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4JX7

Crystal structure of Pim1 kinase in complex with inhibitor 2-[(trans-4-aminocyclohexyl)amino]-4-{[3-(trifluoromethyl)phenyl]amino}pyrido[4,3-d]pyrimidin-5(6H)-one

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1ASerine/threonine-protein kinase pim-1polymer32637293.41UniProt (P11309)
Pfam (PF00069)
In PDB
Homo sapiens (human)Pim1 kinase
2BPIM1 consensus peptidepolymer141592.81Escherichia coli
3A2-[(trans-4-aminocyclohexyl)amino]-4-{[3-(trifluoromethyl)phenyl]amino}pyrido[4,3-d]pyrimidin-5(6H)-onenon-polymer418.41Chemie (1N6)
4waterwater18.0104Chemie (HOH)
Sequence modifications
A: 1 - 313 (UniProt: P11309)
PDBExternal DatabaseDetails
Ala 314-expression tag
Ala 315-expression tag
Ala 316-expression tag
Leu 317-expression tag
Glu 318-expression tag
His 319-expression tag
His 320-expression tag
His 321-expression tag
His 322-expression tag
His 323-expression tag
His 324-expression tag
His 325-expression tag
His 326-expression tag
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains2
Total formula weight38886.3
Non-Polymers*Number of molecules1
Total formula weight418.4
All*Total formula weight39304.7
*Water molecules are not included.

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PDB entries from 2024-09-18

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