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4FJZ

Crystal structure of PI3K-gamma in complex with pyrrolo-pyridine inhibitor 63

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1APhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformpolymer960109824.11UniProt (P48736)
Pfam (PF00794)
Pfam (PF00792)
Pfam (PF00613)
Pfam (PF00454)
In PDB
Homo sapiens (human)PI3-kinase subunit gamma, PI3K-gamma, PI3Kgamma, PtdIns-3-kinase subunit gamma, Phosphatidylinositol 4,5-bisphosphate 3-kinase 110 kDa catalytic subunit gamma, PtdIns-3-kinase subunit p110-gamma, p110gamma, Phosphoinositide-3-kinase catalytic gamma polypeptide, Serine/threonine protein kinase PIK3CG, p120-PI3K
2ASULFATE IONnon-polymer96.14Chemie (SO4)
3A1'-[7-fluoro-3-methyl-2-(pyridin-2-yl)quinolin-4-yl]-6'-(morpholin-4-yl)-1',2,2',3,5,6-hexahydrospiro[pyran-4,3'-pyrrolo[3,2-b]pyridine]non-polymer511.61Chemie (4FJ)
4waterwater18.010Chemie (HOH)
Sequence modifications
A: 144 - 1102 (UniProt: P48736)
PDBExternal DatabaseDetails
Gly 143-expression tag
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains1
Total formula weight109824.1
Non-Polymers*Number of molecules5
Total formula weight895.8
All*Total formula weight110719.9
*Water molecules are not included.

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PDB entries from 2024-06-12

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