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4AP7

Crystal structure of C-MET kinase domain in complex with 4-((6-(4- fluorophenyl)-(1,2,4)triazolo(4,3-b)(1,2,4)triazin-3-yl)methyl)phenol

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1A
(A)
HEPATOCYTE GROWTH FACTOR RECEPTORpolymer30634879.41UniProt (P08581)
Pfam (PF07714)
HOMO SAPIENS (HUMAN)HGF RECEPTOR, HGF/SF RECEPTOR, PROTO-ONCOGENE C-MET, SCATTER FACTOR RECEPTOR, SF RECEPTOR, TYROSINE-PROTEIN KINASE MET
2B
(A)
4-[[6-(4-fluorophenyl)-[1,2,4]triazolo[4,3-b][1,2,4]triazin-3-yl]methyl]phenolnon-polymer321.31Chemie (F47)
3C
(A)
waterwater18.0299Chemie (HOH)
Sequence modifications
A: 1051 - 1348 (UniProt: P08581)
PDBExternal DatabaseDetails
Met 1050-expression tag
His 1349-expression tag
His 1350-expression tag
His 1351-expression tag
His 1352-expression tag
His 1353-expression tag
His 1354-expression tag
His 1355-expression tag
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains1
Total formula weight34879.4
Non-Polymers*Number of molecules1
Total formula weight321.3
All*Total formula weight35200.7
*Water molecules are not included.

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PDB entries from 2025-07-23

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