3ZTX
Aurora kinase selective inhibitors identified using a Taxol-induced checkpoint sensitivity screen.
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | A, B | SERINE/THREONINE-PROTEIN KINASE 12-A | polymer | 284 | 33537.9 | 2 | UniProt (Q6DE08) Pfam (PF00069) In PDB | XENOPUS LAEVIS | AURORA B, AURORA KINASE B-A, AURORA/IPL1-RELATED KINASE 2, A XAIRK2, SERINE/THREONINE-PROTEIN KINASE AURORA-B-A, XAURORA-B |
2 | C, D | INNER CENTROMERE PROTEIN A | polymer | 44 | 5073.8 | 2 | UniProt (O13024) Pfam (PF03941) In PDB | XENOPUS LAEVIS | XL-INCENP, XINC, XINCENP, MITOTIC PHOSPHOPROTEIN 130 |
3 | A, B | 2-((4-(4-HYDROXYPIPERIDIN-1-YL)PHENYL)AMINO)-5,11-DIMETHYL-5H-BENZO[E]PYRIMIDO [5,4-B][1,4]DIAZEPIN-6(11H)-ONE | non-polymer | 430.5 | 2 | Chemie (ZTX) | |||
4 | water | water | 18.0 | 285 | Chemie (HOH) |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 4 |
Total formula weight | 77223.3 | |
Non-Polymers* | Number of molecules | 2 |
Total formula weight | 861.0 | |
All* | Total formula weight | 78084.3 |