3WWJ
Crystal structure of an engineered sitagliptin-producing transaminase, ATA-117-Rd11
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | A, B, C, D, E... | (R)-amine transaminase | polymer | 330 | 36607.1 | 12 | UniProt (F7J696) Pfam (PF01063) In PDB | Arthrobacter sp. KNK168 | R-stereoselective-transaminase |
2 | A, B, C, D, E... | PYRIDOXAL-5'-PHOSPHATE | non-polymer | 247.1 | 12 | Chemie (PLP) | |||
3 | water | water | 18.0 | 1802 | Chemie (HOH) |
Sequence modifications
A, B, C, D, E, F, G, H, I, J, K, L: 1 - 330 (UniProt: F7J696)
PDB | External Database | Details |
---|---|---|
Pro 8 | Ser 8 | ENGINEERED MUTATION |
Phe 60 | Tyr 60 | ENGINEERED MUTATION |
Tyr 61 | Leu 61 | ENGINEERED MUTATION |
Thr 62 | His 62 | ENGINEERED MUTATION |
Ala 65 | Val 65 | ENGINEERED MUTATION |
Thr 69 | Val 69 | ENGINEERED MUTATION |
Gly 81 | Asp 81 | ENGINEERED MUTATION |
Ile 94 | Met 94 | ENGINEERED MUTATION |
Leu 96 | Ile 96 | ENGINEERED MUTATION |
Met 122 | Phe 122 | ENGINEERED MUTATION |
Thr 124 | Ser 124 | ENGINEERED MUTATION |
Thr 126 | Ser 126 | ENGINEERED MUTATION |
Phe 136 | Gly 136 | ENGINEERED MUTATION |
Ser 150 | Tyr 150 | ENGINEERED MUTATION |
Cso 152 | Val 152 | ENGINEERED MUTATION |
Leu 169 | Ala 169 | ENGINEERED MUTATION |
Ile 199 | Val 199 | ENGINEERED MUTATION |
Leu 209 | Ala 209 | ENGINEERED MUTATION |
Cys 215 | Gly 215 | ENGINEERED MUTATION |
Asn 217 | Gly 217 | ENGINEERED MUTATION |
Pro 223 | Ser 223 | ENGINEERED MUTATION |
Pro 269 | Leu 269 | ENGINEERED MUTATION |
Tyr 273 | Leu 273 | ENGINEERED MUTATION |
Ser 282 | Thr 282 | ENGINEERED MUTATION |
Gly 284 | Ala 284 | ENGINEERED MUTATION |
Ser 297 | Pro 297 | ENGINEERED MUTATION |
Val 306 | Ile 306 | ENGINEERED MUTATION |
Pro 321 | Ser 321 | ENGINEERED MUTATION |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 12 |
Total formula weight | 439284.6 | |
Non-Polymers* | Number of molecules | 12 |
Total formula weight | 2965.7 | |
All* | Total formula weight | 442250.3 |