3RFM
Thermostabilised adenosine A2A receptor in complex with caffeine
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | A | Adenosine receptor A2a | polymer | 329 | 36479.1 | 1 | UniProt (P29274) Pfam (PF00001) In PDB | Homo sapiens (human) | |
2 | A | CAFFEINE | non-polymer | 194.2 | 1 | Chemie (CFF) |
Sequence modifications
A: 1 - 317 (UniProt: P29274)
PDB | External Database | Details |
---|---|---|
Leu 54 | Ala 54 | engineered mutation |
Ala 88 | Thr 88 | engineered mutation |
Ala 107 | Arg 107 | engineered mutation |
Ala 122 | Lys 122 | engineered mutation |
Ala 202 | Leu 202 | engineered mutation |
Ala 235 | Leu 235 | engineered mutation |
Ala 239 | Val 239 | engineered mutation |
Ala 277 | Ser 277 | engineered mutation |
Ala 318 | - | expression tag |
Ala 319 | - | expression tag |
His 320 | - | expression tag |
His 321 | - | expression tag |
His 322 | - | expression tag |
His 323 | - | expression tag |
His 324 | - | expression tag |
His 325 | - | expression tag |
His 326 | - | expression tag |
His 327 | - | expression tag |
His 328 | - | expression tag |
His 329 | - | expression tag |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 1 |
Total formula weight | 36479.1 | |
Non-Polymers* | Number of molecules | 1 |
Total formula weight | 194.2 | |
All* | Total formula weight | 36673.3 |