3ETA
Kinase domain of insulin receptor complexed with a pyrrolo pyridine inhibitor
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | A, B | insulin receptor, kinase domain | polymer | 317 | 36156.3 | 2 | UniProt (P06213) Pfam (PF07714) In PDB | Homo sapiens (human) | IR, Insulin receptor subunit alpha, Insulin receptor subunit beta |
2 | A, B | 1-(3-{5-[4-(aminomethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-3-yl}phenyl)-3-(2-phenoxyphenyl)urea | non-polymer | 525.6 | 2 | Chemie (351) | |||
3 | water | water | 18.0 | 210 | Chemie (HOH) |
Sequence modifications
A, B: 990 - 1295 (UniProt: P06213)
PDB | External Database | Details |
---|---|---|
Met 979 | - | expression tag |
Lys 980 | - | expression tag |
Lys 981 | - | expression tag |
Gly 982 | - | expression tag |
His 983 | - | expression tag |
His 984 | - | expression tag |
His 985 | - | expression tag |
His 986 | - | expression tag |
His 987 | - | expression tag |
His 988 | - | expression tag |
Gly 989 | - | expression tag |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 2 |
Total formula weight | 72312.6 | |
Non-Polymers* | Number of molecules | 2 |
Total formula weight | 1051.2 | |
All* | Total formula weight | 73363.8 |