3C7Q
Structure of VEGFR2 kinase domain in complex with BIBF1120
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | A | Vascular endothelial growth factor receptor 2 | polymer | 316 | 36557.0 | 1 | UniProt (P35968) Pfam (PF07714) In PDB | Homo sapiens (Human) | VEGFR-2, Kinase insert domain receptor, Protein-tyrosine kinase receptor Flk-1, CD309 antigen |
2 | A | SULFATE ION | non-polymer | 96.1 | 5 | Chemie (SO4) | |||
3 | A | methyl (3Z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1H-indole-6-carboxylate | non-polymer | 539.6 | 1 | Chemie (XIN) | |||
4 | water | water | 18.0 | 206 | Chemie (HOH) |
Sequence modifications
A: 806 - 1171 (UniProt: P35968)
PDB | External Database | Details |
---|---|---|
Gly 804 | - | expression tag |
Ser 805 | - | expression tag |
- | Thr 940 | deletion |
- | Lys 941 | deletion |
- | Gly 942 | deletion |
- | Ala 943 | deletion |
- | Arg 944 | deletion |
- | Phe 945 | deletion |
- | Arg 946 | deletion |
- | Gln 947 | deletion |
- | Gly 948 | deletion |
- | Lys 949 | deletion |
- | Asp 950 | deletion |
- | Tyr 951 | deletion |
- | Val 952 | deletion |
- | Gly 953 | deletion |
- | Ala 954 | deletion |
- | Ile 955 | deletion |
- | Pro 956 | deletion |
- | Val 957 | deletion |
- | Asp 958 | deletion |
- | Leu 959 | deletion |
- | Lys 960 | deletion |
- | Arg 961 | deletion |
- | Arg 962 | deletion |
- | Leu 963 | deletion |
- | Asp 964 | deletion |
- | Ser 965 | deletion |
- | Ile 966 | deletion |
- | Thr 967 | deletion |
- | Ser 968 | deletion |
- | Ser 969 | deletion |
- | Gln 970 | deletion |
- | Ser 971 | deletion |
- | Ser 972 | deletion |
- | Ala 973 | deletion |
- | Ser 974 | deletion |
- | Ser 975 | deletion |
- | Gly 976 | deletion |
- | Phe 977 | deletion |
- | Val 978 | deletion |
- | Glu 979 | deletion |
- | Glu 980 | deletion |
- | Lys 981 | deletion |
- | Ser 982 | deletion |
- | Leu 983 | deletion |
- | Ser 984 | deletion |
- | Asp 985 | deletion |
- | Val 986 | deletion |
- | Glu 987 | deletion |
- | Glu 988 | deletion |
- | Glu 989 | deletion |
- | Glu 990 | deletion |
- | Ala 991 | deletion |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 1 |
Total formula weight | 36557.0 | |
Non-Polymers* | Number of molecules | 6 |
Total formula weight | 1019.9 | |
All* | Total formula weight | 37576.9 |