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2Y00

TURKEY BETA1 ADRENERGIC RECEPTOR WITH STABILISING MUTATIONS AND BOUND PARTIAL AGONIST DOBUTAMINE (CRYSTAL DOB92)

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1A, BBETA-1 ADRENERGIC RECEPTORpolymer31535940.82UniProt (P07700)
Pfam (PF00001)
In PDB
MELEAGRIS GALLOPAVO (TURKEY)BETA-1 ADRENORECEPTOR, BETA-1 ADRENOCEPTOR, BETA-T
2A, BCHOLESTEROL HEMISUCCINATEnon-polymer486.74Chemie (Y01)
3A, BHEGA-10non-polymer379.510Chemie (2CV)
4A, BDOBUTAMINEnon-polymer301.42Chemie (Y00)
5ASODIUM IONnon-polymer23.01Chemie (NA)
6waterwater18.038Chemie (HOH)
Sequence modifications
A, B: 33 - 368 (UniProt: P07700)
PDBExternal DatabaseDetails
Met 31-expression tag
Gly 32-expression tag
Ser 68Arg 68engineered mutation
Val 90Met 90engineered mutation
Leu 116Cys 116engineered mutation
Ala 227Tyr 227engineered mutation
-Cys 244deletion
-Glu 245deletion
-Gly 246deletion
-Arg 247deletion
-Phe 248deletion
-Tyr 249deletion
-Gly 250deletion
-Ser 251deletion
-Gln 252deletion
-Glu 253deletion
-Gln 254deletion
-Pro 255deletion
-Gln 256deletion
-Pro 257deletion
-Pro 258deletion
-Pro 259deletion
-Leu 260deletion
-Pro 261deletion
-Gln 262deletion
-His 263deletion
-Gln 264deletion
-Pro 265deletion
-Ile 266deletion
-Leu 267deletion
-Gly 268deletion
-Asn 269deletion
-Gly 270deletion
-Arg 271deletion
Leu 282Ala 282engineered mutation
Ala 327Phe 327engineered mutation
Met 338Phe 338engineered mutation
Ala 358Cys 358engineered mutation
His 369-expression tag
His 370-expression tag
His 371-expression tag
His 372-expression tag
His 373-expression tag
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains2
Total formula weight71881.6
Non-Polymers*Number of molecules17
Total formula weight6367.5
All*Total formula weight78249.1
*Water molecules are not included.

217705

PDB entries from 2024-03-27

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