2VX1
ephB4 kinase domain inhibitor complex
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | A | EPHRIN TYPE-B RECEPTOR 4 | polymer | 302 | 33934.8 | 1 | UniProt (P54760) Pfam (PF07714) In PDB | HOMO SAPIENS (HUMAN) | TYROSINE-PROTEIN KINASE RECEPTOR HTK, TYROSINE-PROTEIN KINASE TYRO11, EPHB4 RECEPTOR TYROSINE KINASE |
2 | A | 3-({4-[(5-CHLORO-1,3-BENZODIOXOL-4-YL)AMINO]PYRIMIDIN-2-YL}AMINO)BENZAMIDE | non-polymer | 383.8 | 1 | Chemie (7X8) | |||
3 | A | MAGNESIUM ION | non-polymer | 24.3 | 3 | Chemie (MG) | |||
4 | water | water | 18.0 | 260 | Chemie (HOH) |
Sequence modifications
A: 598 - 899 (UniProt: P54760)
PDB | External Database | Details |
---|---|---|
Glu 774 | Tyr 774 | engineered mutation |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 1 |
Total formula weight | 33934.8 | |
Non-Polymers* | Number of molecules | 4 |
Total formula weight | 456.7 | |
All* | Total formula weight | 34391.5 |