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2JAV

Human Kinase with pyrrole-indolinone ligand

Replaces:  2CL1
Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1A
(A)
SERINE/THREONINE-PROTEIN KINASE NEK2polymer27932632.51UniProt (P51955)
Pfam (PF00069)
HOMO SAPIENS (HUMAN)NIMA-RELATED PROTEIN KINASE 2, NIMA-LIKE PROTEIN KINASE 1, HSPK 21, NEVER IN MITOSIS GENE A-RELATED KINASE 2
2B
(A)
5-[(Z)-(5-CHLORO-2-OXO-1,2-DIHYDRO-3H-INDOL-3-YLIDENE)METHYL]-N-(DIETHYLAMINO)ETHYL]-2,4-DIMETHYL-1H-PYRROLE-3-CARBOXAMIDEnon-polymer329.81Chemie (5Z5)
3C
(A)
waterwater18.0107Chemie (HOH)
Sequence modifications
A: 1 - 271 (UniProt: P51955)
PDBExternal DatabaseDetails
Ala 175Thr 175engineered mutation
A: 272 - 279 (PDB: 2JAV)
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains1
Total formula weight32632.5
Non-Polymers*Number of molecules1
Total formula weight329.8
All*Total formula weight32962.2
*Water molecules are not included.

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PDB entries from 2025-06-18

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