2I1M
cFMS tyrosine kinase (tie2 KID) in complex with an arylamide inhibitor
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | A | Macrophage colony-stimulating factor 1 receptor | polymer | 333 | 37613.1 | 1 | UniProt (P07333) Pfam (PF07714) In PDB | Homo sapiens (human) | cFMS Receptor Tyrosine Kinase, CSF-1-R, Fms proto-oncogene, c-fms, CD115 antigen |
2 | A | 5-CYANO-FURAN-2-CARBOXYLIC ACID [5-HYDROXYMETHYL-2-(4-METHYL-PIPERIDIN-1-YL)-PHENYL]-AMIDE | non-polymer | 339.4 | 1 | Chemie (5CN) | |||
3 | water | water | 18.0 | 176 | Chemie (HOH) |
Sequence modifications
A: 538 - 678 (UniProt: P07333)
A: 753 - 922 (UniProt: P07333)
PDB | External Database | Details |
---|---|---|
Gly 535 | - | expression tag |
Val 536 | - | expression tag |
Asp 537 | - | expression tag |
PDB | External Database | Details |
---|---|---|
Ser 679 | - | SEE REMARK 999 |
Arg 680 | - | SEE REMARK 999 |
Val 681 | - | SEE REMARK 999 |
Leu 682 | - | SEE REMARK 999 |
Glu 683 | - | SEE REMARK 999 |
Thr 684 | - | SEE REMARK 999 |
Asp 685 | - | SEE REMARK 999 |
Pro 686 | - | SEE REMARK 999 |
Ala 687 | - | SEE REMARK 999 |
Phe 688 | - | SEE REMARK 999 |
Ala 689 | - | SEE REMARK 999 |
Ile 690 | - | SEE REMARK 999 |
Ala 691 | - | SEE REMARK 999 |
Asn 692 | - | SEE REMARK 999 |
Ser 693 | - | SEE REMARK 999 |
Thr 694 | - | SEE REMARK 999 |
Ala 697 | - | SEE REMARK 999 |
Ser 698 | - | SEE REMARK 999 |
Thr 699 | - | SEE REMARK 999 |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 1 |
Total formula weight | 37613.1 | |
Non-Polymers* | Number of molecules | 1 |
Total formula weight | 339.4 | |
All* | Total formula weight | 37952.5 |