2I0V
c-FMS tyrosine kinase in complex with a quinolone inhibitor
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | A | cFMS tyrosine kinase | polymer | 335 | 38064.5 | 1 | UniProt (P07333) Pfam (PF07714) In PDB | Homo sapiens (human) | |
2 | A | SULFATE ION | non-polymer | 96.1 | 1 | Chemie (SO4) | |||
3 | A | 6-CHLORO-3-(3-METHYLISOXAZOL-5-YL)-4-PHENYLQUINOLIN-2(1H)-ONE | non-polymer | 336.8 | 1 | Chemie (6C3) | |||
4 | water | water | 18.0 | 26 | Chemie (HOH) |
Sequence modifications
A: 538 - 678 (UniProt: P07333)
A: 753 - 922 (UniProt: P07333)
PDB | External Database | Details |
---|---|---|
Gly 535 | - | expression tag |
Val 536 | - | expression tag |
Asp 537 | - | expression tag |
PDB | External Database | Details |
---|---|---|
Arg 679 | - | SEE REMARK 999 |
Pro 680 | - | SEE REMARK 999 |
Pro 681 | - | SEE REMARK 999 |
Gly 682 | - | SEE REMARK 999 |
Leu 683 | - | SEE REMARK 999 |
Glu 684 | - | SEE REMARK 999 |
Tyr 685 | - | SEE REMARK 999 |
Ser 686 | - | SEE REMARK 999 |
Tyr 687 | - | SEE REMARK 999 |
Asn 688 | - | SEE REMARK 999 |
Pro 689 | - | SEE REMARK 999 |
Ser 690 | - | SEE REMARK 999 |
His 691 | - | SEE REMARK 999 |
Asn 692 | - | SEE REMARK 999 |
Pro 693 | - | SEE REMARK 999 |
Glu 694 | - | SEE REMARK 999 |
Glu 695 | - | SEE REMARK 999 |
Gln 696 | - | SEE REMARK 999 |
Leu 697 | - | SEE REMARK 999 |
Ser 698 | - | SEE REMARK 999 |
Ser 699 | - | SEE REMARK 999 |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 1 |
Total formula weight | 38064.5 | |
Non-Polymers* | Number of molecules | 2 |
Total formula weight | 432.8 | |
All* | Total formula weight | 38497.3 |