1OGU
STRUCTURE OF HUMAN THR160-PHOSPHO CDK2/CYCLIN A COMPLEXED WITH A 2-ARYLAMINO-4-CYCLOHEXYLMETHYL-5-NITROSO-6-AMINOPYRIMIDINE INHIBITOR
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | A, C | CELL DIVISION PROTEIN KINASE 2 | polymer | 302 | 34354.8 | 2 | UniProt (P24941) Pfam (PF00069) In PDB | HOMO SAPIENS (HUMAN) | P33 PROTEIN KINASE |
2 | B, D | CYCLIN A2 | polymer | 260 | 29884.6 | 2 | UniProt (P20248) Pfam (PF00134) Pfam (PF02984) In PDB | HOMO SAPIENS (HUMAN) | CYCLIN A, CYCLIN A3 |
3 | A, C | 4-{[4-AMINO-6-(CYCLOHEXYLMETHOXY)-5-NITROSOPYRIMIDIN-2-YL]AMINO}BENZAMIDE | non-polymer | 370.4 | 2 | Chemie (ST8) | |||
4 | B, D | MONOTHIOGLYCEROL | non-polymer | 108.2 | 2 | Chemie (SGM) | |||
5 | water | water | 18.0 | 134 | Chemie (HOH) |
Sequence modifications
A, C: -3 - 0 (PDB: 1OGU)
A, C: 1 - 298 (UniProt: P24941)
B, D: 173 - 173 (PDB: 1OGU)
B, D: 174 - 432 (UniProt: P20248)
A, C: 1 - 298 (UniProt: P24941)
B, D: 173 - 173 (PDB: 1OGU)
B, D: 174 - 432 (UniProt: P20248)
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 4 |
Total formula weight | 128478.8 | |
Non-Polymers* | Number of molecules | 4 |
Total formula weight | 957.1 | |
All* | Total formula weight | 129435.9 |