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1GWQ

HUMAN OESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH RALOXIFENE CORE AND TIF2 NRBOX2 PEPTIDE

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1A, B
(A, B)
OESTROGEN RECEPTORpolymer24828368.42UniProt (P03372)
Pfam (PF00104)
HOMO SAPIENS (HUMAN)ER, ESTRADIOL RECEPTOR, ER-ALPHA
2C, D
(C, D)
NUCLEAR RECEPTOR COACTIVATOR 2polymer91138.42UniProt (Q15596)HOMO SAPIENSTRANSCRIPTION INTERMEDIARY FACTOR-2, TIF2
3E, F
(A, B)
RALOXIFENE COREnon-polymer242.32Chemie (ZTW)
4G, H
(A, B)
waterwater18.0119Chemie (HOH)
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains4
Total formula weight59013.6
Non-Polymers*Number of molecules2
Total formula weight484.6
All*Total formula weight59498.2
*Water molecules are not included.

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PDB entries from 2025-06-11

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