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1C5M

STRUCTURAL BASIS FOR SELECTIVITY OF A SMALL MOLECULE, S1-BINDING, SUB-MICROMOLAR INHIBITOR OF UROKINASE TYPE PLASMINOGEN ACTIVATOR

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1A
(D)
PROTEIN (COAGULATION FACTOR X)polymer25528649.71UniProt (P00742)
Pfam (PF00089)
Homo sapiens (human)
2B
(F)
PROTEIN (COAGULATION FACTOR X)polymer9610533.71UniProt (P00742)
Pfam (PF00008)
Pfam (PF14670)
Homo sapiens (human)
3C, D
(D, F)
waterwater18.0454Chemie (HOH)
Sequence modifications
D: 16 - 265 (UniProt: P00742)
PDBExternal DatabaseDetails
Val 257-insertion
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains2
Total formula weight39183.4
All*Total formula weight39183.4
*Water molecules are not included.

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PDB entries from 2025-06-11

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