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9H2X

Crystal structure of stabilized A2A adenosine receptor A2AR-StaR2-bRIL in complex with compound 7, a novel nanomolar A2A receptor antagonist from modern hit-finding with structure-guided de novo design

This is a non-PDB format compatible entry.
Resources
File formatFile name (file size)
PDBx/mmCIF9h2x.cif.gz Display(192.58 KB)
9h2x.cif
PDBx/mmJSONall9h2x.json.gz Display (Tree)(134.28 KB)
9h2x.json
no-atom9h2x-noatom.json.gz Display (Header)(21.28 KB)
9h2x-noatom.json
add only9h2x-plus.json.gz Display(400.00 B)
9h2x-plus.json
PDBMLall9h2x.xml.gz Display(256.34 KB)
9h2x.xml
no-atom9h2x-noatom.xml.gz Display(36.59 KB)
9h2x-noatom.xml
ext-atom9h2x-extatom.xml.gz Display(80.44 KB)
9h2x-extatom.xml
RDF9h2x.rdf.gz Visualize(102.61 KB)
9h2x.rdf
Structure factorsr9h2xsf.ent.gz Display(47.93 MB)
r9h2xsf.ent
Biological unit (mmCIF format)9h2x-assembly1.cif.gz Display(176.61 KB)
9h2x-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF9h2x_validation.pdf.gz Display(3.70 MB)
9h2x_validation.pdf
PDF-full9h2x_full_validation.pdf.gz Display(3.81 MB)
9h2x_full_validation.pdf
mmCIF9h2x_validation.cif.gz Display(28.18 KB)
9h2x_validation.cif
XML9h2x_validation.xml.gz Display(21.15 KB)
9h2x_validation.xml
PNG9h2x_multipercentile_validation.png.gz Display(165.52 KB)
9h2x_multipercentile_validation.png
SVG9h2x_multipercentile_validation.svg.gz Display(957.00 B)
9h2x_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)9h2x_validation_2fo-fc_map_coef.cif.gz Display(676.28 KB)
9h2x_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)9h2x_validation_fo-fc_map_coef.cif.gz Display(672.82 KB)
9h2x_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)9h2x_validation_2fo-fc_map_coef.mtz Visualize(1.17 MB)
fo-fc (MTZ)9h2x_validation_fo-fc_map_coef.mtz Visualize(1.17 MB)

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PDB entries from 2025-06-18

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