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8U0Q

Co-crystal structure of optimized analog TDI-13537 provided new insights into the potency determinants of the sulfonamide inhibitor series

Resources
File formatFile name (file size)
PDBx/mmCIF8u0q.cif.gz Display(255.21 KB)
8u0q.cif
PDBx/mmJSONall8u0q.json.gz Display (Tree)(179.34 KB)
8u0q.json
no-atom8u0q-noatom.json.gz Display (Header)(22.63 KB)
8u0q-noatom.json
add only8u0q-plus.json.gz Display(1.37 KB)
8u0q-plus.json
PDBMLall8u0q.xml.gz Display(324.69 KB)
8u0q.xml
no-atom8u0q-noatom.xml.gz Display(47.27 KB)
8u0q-noatom.xml
ext-atom8u0q-extatom.xml.gz Display(219.91 KB)
8u0q-extatom.xml
PDBpdb8u0q.ent.gz Display(164.10 KB)
pdb8u0q.ent
RDF8u0q.rdf.gz Visualize(133.00 KB)
8u0q.rdf
Structure factorsr8u0qsf.ent.gz Display(4.42 MB)
r8u0qsf.ent
Biological unit (mmCIF format)8u0q-assembly1.cif.gz Display(212.86 KB)
8u0q-assembly1.cif (A,B)

*author and software defined assembly, 2 molecule(s) (dimeric)

Biological unit (PDB format)8u0q.pdb1.gz Display(156.43 KB)
8u0q.pdb1 (A,B)

*author and software defined assembly, 2 molecule(s) (dimeric)

Validation reportsPDF8u0q_validation.pdf.gz Display(1.38 MB)
8u0q_validation.pdf
PDF-full8u0q_full_validation.pdf.gz Display(1.41 MB)
8u0q_full_validation.pdf
mmCIF8u0q_validation.cif.gz Display(61.24 KB)
8u0q_validation.cif
XML8u0q_validation.xml.gz Display(41.87 KB)
8u0q_validation.xml
PNG8u0q_multipercentile_validation.png.gz Display(161.21 KB)
8u0q_multipercentile_validation.png
SVG8u0q_multipercentile_validation.svg.gz Display(955.00 B)
8u0q_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)8u0q_validation_2fo-fc_map_coef.cif.gz Display(1.09 MB)
8u0q_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)8u0q_validation_fo-fc_map_coef.cif.gz Display(1.06 MB)
8u0q_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)8u0q_validation_2fo-fc_map_coef.mtz Visualize(2.61 MB)
fo-fc (MTZ)8u0q_validation_fo-fc_map_coef.mtz Visualize(2.61 MB)

222036

PDB entries from 2024-07-03

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