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8G3E

Crystal structure of human WDR5 in complex with (1M)-N-[(3,5-difluoro[1,1'-biphenyl]-4-yl)methyl]-6-methyl-4-oxo-1-(pyridin-3-yl)-1,4-dihydropyridazine-3-carboxamide (compound 2, WDR5-MYC inhibitor)

Resources
File formatFile name (file size)
PDBx/mmCIF8g3e.cif.gz Display(276.46 KB)
8g3e.cif
PDBx/mmJSONall8g3e.json.gz Display (Tree)(189.99 KB)
8g3e.json
no-atom8g3e-noatom.json.gz Display (Header)(18.16 KB)
8g3e-noatom.json
add only8g3e-plus.json.gz Display(1.56 KB)
8g3e-plus.json
PDBMLall8g3e.xml.gz Display(384.74 KB)
8g3e.xml
no-atom8g3e-noatom.xml.gz Display(35.99 KB)
8g3e-noatom.xml
ext-atom8g3e-extatom.xml.gz Display(120.89 KB)
8g3e-extatom.xml
PDBpdb8g3e.ent.gz Display(221.32 KB)
pdb8g3e.ent
RDF8g3e.rdf.gz Visualize(101.95 KB)
8g3e.rdf
Structure factorsr8g3esf.ent.gz Display(3.23 MB)
r8g3esf.ent
Biological unit (mmCIF format)8g3e-assembly1.cif.gz Display(138.23 KB)
8g3e-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

8g3e-assembly2.cif.gz Display(138.06 KB)
8g3e-assembly2.cif (B)

*author defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)8g3e.pdb1.gz Display(109.69 KB)
8g3e.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

8g3e.pdb2.gz Display(110.65 KB)
8g3e.pdb2 (B)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF8g3e_validation.pdf.gz Display(965.65 KB)
8g3e_validation.pdf
PDF-full8g3e_full_validation.pdf.gz Display(971.30 KB)
8g3e_full_validation.pdf
mmCIF8g3e_validation.cif.gz Display(45.27 KB)
8g3e_validation.cif
XML8g3e_validation.xml.gz Display(29.92 KB)
8g3e_validation.xml
PNG8g3e_multipercentile_validation.png.gz Display(156.87 KB)
8g3e_multipercentile_validation.png
SVG8g3e_multipercentile_validation.svg.gz Display(922.00 B)
8g3e_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)8g3e_validation_2fo-fc_map_coef.cif.gz Display(1.34 MB)
8g3e_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)8g3e_validation_fo-fc_map_coef.cif.gz Display(1.25 MB)
8g3e_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)8g3e_validation_2fo-fc_map_coef.mtz Visualize(3.22 MB)
fo-fc (MTZ)8g3e_validation_fo-fc_map_coef.mtz Visualize(3.22 MB)

221371

PDB entries from 2024-06-19

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