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8DI4

Discovery of MK-8189, a highly potent and selective PDE10A inhibitor for the treatment of schizophrenia

Resources
File formatFile name (file size)
PDBx/mmCIF8di4.cif.gz Display(145.12 KB)
8di4.cif
PDBx/mmJSONall8di4.json.gz Display (Tree)(94.68 KB)
8di4.json
no-atom8di4-noatom.json.gz Display (Header)(17.62 KB)
8di4-noatom.json
add only8di4-plus.json.gz Display(986.00 B)
8di4-plus.json
PDBMLall8di4.xml.gz Display(192.82 KB)
8di4.xml
no-atom8di4-noatom.xml.gz Display(34.61 KB)
8di4-noatom.xml
ext-atom8di4-extatom.xml.gz Display(119.56 KB)
8di4-extatom.xml
pdb_nextgenallpdb_00008di4_xyz-enrich.cif.gz Display(158.75 KB)
pdb_00008di4_xyz-enrich.cif
no-atompdb_00008di4_xyz-no-atom-enrich.xml.gz Display(43.04 KB)
pdb_00008di4_xyz-no-atom-enrich.xml
ng-only8di4-plus.json.gz Display(3.21 KB)
8di4-plus.json
PDBpdb8di4.ent.gz Display(111.75 KB)
pdb8di4.ent
RDF8di4.rdf.gz Visualize(100.70 KB)
8di4.rdf
Structure factorsr8di4sf.ent.gz Display(2.43 MB)
r8di4sf.ent
Biological unit (mmCIF format)8di4-assembly1.cif.gz Display(70.30 KB)
8di4-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

8di4-assembly2.cif.gz Display(69.84 KB)
8di4-assembly2.cif (B)

*author defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)8di4.pdb1.gz Display(54.67 KB)
8di4.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

8di4.pdb2.gz Display(54.75 KB)
8di4.pdb2 (B)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF8di4_validation.pdf.gz Display(917.03 KB)
8di4_validation.pdf
PDF-full8di4_full_validation.pdf.gz Display(922.49 KB)
8di4_full_validation.pdf
mmCIF8di4_validation.cif.gz Display(34.41 KB)
8di4_validation.cif
XML8di4_validation.xml.gz Display(24.61 KB)
8di4_validation.xml
PNG8di4_multipercentile_validation.png.gz Display(170.64 KB)
8di4_multipercentile_validation.png
SVG8di4_multipercentile_validation.svg.gz Display(976.00 B)
8di4_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)8di4_validation_2fo-fc_map_coef.cif.gz Display(424.90 KB)
8di4_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)8di4_validation_fo-fc_map_coef.cif.gz Display(413.24 KB)
8di4_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)8di4_validation_2fo-fc_map_coef.mtz Visualize(1014.64 KB)
fo-fc (MTZ)8di4_validation_fo-fc_map_coef.mtz Visualize(1014.64 KB)

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PDB entries from 2026-02-11

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