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7UAS

Discovery of Potent Orally Bioavailable WD Repeat Domain 5 (WDR5) Inhibitors Using a Pharmacophore-Based Optimization

Resources
File formatFile name (file size)
PDBx/mmCIF7uas.cif.gz Display(255.60 KB)
7uas.cif
PDBx/mmJSONall7uas.json.gz Display (Tree)(171.88 KB)
7uas.json
no-atom7uas-noatom.json.gz Display (Header)(19.51 KB)
7uas-noatom.json
add only7uas-plus.json.gz Display(1.64 KB)
7uas-plus.json
PDBMLall7uas.xml.gz Display(353.81 KB)
7uas.xml
no-atom7uas-noatom.xml.gz Display(39.14 KB)
7uas-noatom.xml
ext-atom7uas-extatom.xml.gz Display(118.88 KB)
7uas-extatom.xml
pdb_nextgenallpdb_00007uas_xyz-enrich.cif.gz Display(268.48 KB)
pdb_00007uas_xyz-enrich.cif
no-atompdb_00007uas_xyz-no-atom-enrich.xml.gz Display(47.19 KB)
pdb_00007uas_xyz-no-atom-enrich.xml
ng-only7uas-plus.json.gz Display(2.29 KB)
7uas-plus.json
PDBpdb7uas.ent.gz Display(202.63 KB)
pdb7uas.ent
RDF7uas.rdf.gz Visualize(107.51 KB)
7uas.rdf
Structure factorsr7uassf.ent.gz Display(1.23 MB)
r7uassf.ent
Biological unit (mmCIF format)7uas-assembly1.cif.gz Display(126.05 KB)
7uas-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

7uas-assembly2.cif.gz Display(127.20 KB)
7uas-assembly2.cif (B)

*author defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)7uas.pdb1.gz Display(99.54 KB)
7uas.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

7uas.pdb2.gz Display(100.72 KB)
7uas.pdb2 (B)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF7uas_validation.pdf.gz Display(1.22 MB)
7uas_validation.pdf
PDF-full7uas_full_validation.pdf.gz Display(1.23 MB)
7uas_full_validation.pdf
mmCIF7uas_validation.cif.gz Display(46.01 KB)
7uas_validation.cif
XML7uas_validation.xml.gz Display(30.34 KB)
7uas_validation.xml
PNG7uas_multipercentile_validation.png.gz Display(161.36 KB)
7uas_multipercentile_validation.png
SVG7uas_multipercentile_validation.svg.gz Display(949.00 B)
7uas_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)7uas_validation_2fo-fc_map_coef.cif.gz Display(503.12 KB)
7uas_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)7uas_validation_fo-fc_map_coef.cif.gz Display(478.08 KB)
7uas_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)7uas_validation_2fo-fc_map_coef.mtz Visualize(1.18 MB)
fo-fc (MTZ)7uas_validation_fo-fc_map_coef.mtz Visualize(1.18 MB)

246905

PDB entries from 2025-12-31

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