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7U8H

Discovery of a KRAS G12V Inhibitor in vivo Tool Compound starting from an HSQC-NMR based Fragment Hit

Resources
File formatFile name (file size)
PDBx/mmCIF7u8h.cif.gz Display(308.31 KB)
7u8h.cif
PDBx/mmJSONall7u8h.json.gz Display (Tree)(203.88 KB)
7u8h.json
no-atom7u8h-noatom.json.gz Display (Header)(22.06 KB)
7u8h-noatom.json
add only7u8h-plus.json.gz Display(1.06 KB)
7u8h-plus.json
PDBMLall7u8h.xml.gz Display(425.50 KB)
7u8h.xml
no-atom7u8h-noatom.xml.gz Display(45.44 KB)
7u8h-noatom.xml
ext-atom7u8h-extatom.xml.gz Display(141.73 KB)
7u8h-extatom.xml
PDBpdb7u8h.ent.gz Display(250.79 KB)
pdb7u8h.ent
RDF7u8h.rdf.gz Visualize(115.13 KB)
7u8h.rdf
Structure factorsr7u8hsf.ent.gz Display(1.88 MB)
r7u8hsf.ent
Biological unit (mmCIF format)7u8h-assembly1.cif.gz Display(79.96 KB)
7u8h-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

7u8h-assembly2.cif.gz Display(78.86 KB)
7u8h-assembly2.cif (B)

*author and software defined assembly, 1 molecule(s) (monomeric)

7u8h-assembly3.cif.gz Display(74.26 KB)
7u8h-assembly3.cif (C)

*author and software defined assembly, 1 molecule(s) (monomeric)

7u8h-assembly4.cif.gz Display(80.87 KB)
7u8h-assembly4.cif (D)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)7u8h.pdb1.gz Display(63.95 KB)
7u8h.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

7u8h.pdb2.gz Display(62.79 KB)
7u8h.pdb2 (B)

*author and software defined assembly, 1 molecule(s) (monomeric)

7u8h.pdb3.gz Display(58.48 KB)
7u8h.pdb3 (C)

*author and software defined assembly, 1 molecule(s) (monomeric)

7u8h.pdb4.gz Display(64.27 KB)
7u8h.pdb4 (D)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF7u8h_validation.pdf.gz Display(2.39 MB)
7u8h_validation.pdf
PDF-full7u8h_full_validation.pdf.gz Display(2.40 MB)
7u8h_full_validation.pdf
mmCIF7u8h_validation.cif.gz Display(50.34 KB)
7u8h_validation.cif
XML7u8h_validation.xml.gz Display(35.36 KB)
7u8h_validation.xml
PNG7u8h_multipercentile_validation.png.gz Display(166.76 KB)
7u8h_multipercentile_validation.png
SVG7u8h_multipercentile_validation.svg.gz Display(977.00 B)
7u8h_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)7u8h_validation_2fo-fc_map_coef.cif.gz Display(764.20 KB)
7u8h_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)7u8h_validation_fo-fc_map_coef.cif.gz Display(748.06 KB)
7u8h_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)7u8h_validation_2fo-fc_map_coef.mtz Visualize(1.76 MB)
fo-fc (MTZ)7u8h_validation_fo-fc_map_coef.mtz Visualize(1.76 MB)

222415

PDB entries from 2024-07-10

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