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7KSI

Thiophenyl-Pyrazolourea Derivatives as Potent, Brian Penetrant, Orally Bioavailable, and Isoform-Selective JNK3 Inhibitors

Resources
File formatFile name (file size)
PDBx/mmCIF7ksi.cif.gz Display(225.60 KB)
7ksi.cif
PDBx/mmJSONall7ksi.json.gz Display (Tree)(153.77 KB)
7ksi.json
no-atom7ksi-noatom.json.gz Display (Header)(18.94 KB)
7ksi-noatom.json
add only7ksi-plus.json.gz Display(1.21 KB)
7ksi-plus.json
PDBMLall7ksi.xml.gz Display(301.29 KB)
7ksi.xml
no-atom7ksi-noatom.xml.gz Display(31.45 KB)
7ksi-noatom.xml
ext-atom7ksi-extatom.xml.gz Display(130.16 KB)
7ksi-extatom.xml
PDBpdb7ksi.ent.gz Display(181.48 KB)
pdb7ksi.ent
RDF7ksi.rdf.gz Visualize(93.87 KB)
7ksi.rdf
Structure factorsr7ksisf.ent.gz Display(973.91 KB)
r7ksisf.ent
Biological unit (mmCIF format)7ksi-assembly1.cif.gz Display(214.82 KB)
7ksi-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)7ksi.pdb1.gz Display(175.77 KB)
7ksi.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF7ksi_validation.pdf.gz Display(715.01 KB)
7ksi_validation.pdf
PDF-full7ksi_full_validation.pdf.gz Display(717.94 KB)
7ksi_full_validation.pdf
mmCIF7ksi_validation.cif.gz Display(26.50 KB)
7ksi_validation.cif
XML7ksi_validation.xml.gz Display(17.62 KB)
7ksi_validation.xml
PNG7ksi_multipercentile_validation.png.gz Display(172.55 KB)
7ksi_multipercentile_validation.png
SVG7ksi_multipercentile_validation.svg.gz Display(981.00 B)
7ksi_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)7ksi_validation_2fo-fc_map_coef.cif.gz Display(402.33 KB)
7ksi_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)7ksi_validation_fo-fc_map_coef.cif.gz Display(307.68 KB)
7ksi_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)7ksi_validation_2fo-fc_map_coef.mtz Visualize(1004.63 KB)
fo-fc (MTZ)7ksi_validation_fo-fc_map_coef.mtz Visualize(1004.63 KB)

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PDB entries from 2024-07-24

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