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7G2E

Crystal Structure of rat Autotaxin in complex with 2-(3,4-dichlorophenyl)-1-[4-[(4-fluorophenyl)methyl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]ethanone, i.e. SMILES Fc1ccc(cc1)Cc1c2CN(C(=O)Cc3ccc(Cl)c(Cl)c3)CCc2ncn1 with IC50=0.795943 microM

Resources
File formatFile name (file size)
PDBx/mmCIF7g2e.cif.gz Display(200.93 KB)
7g2e.cif
PDBx/mmJSONall7g2e.json.gz Display (Tree)(135.62 KB)
7g2e.json
no-atom7g2e-noatom.json.gz Display (Header)(27.68 KB)
7g2e-noatom.json
add only7g2e-plus.json.gz Display(1.94 KB)
7g2e-plus.json
PDBMLall7g2e.xml.gz Display(268.41 KB)
7g2e.xml
no-atom7g2e-noatom.xml.gz Display(52.60 KB)
7g2e-noatom.xml
ext-atom7g2e-extatom.xml.gz Display(163.17 KB)
7g2e-extatom.xml
pdb_nextgenallpdb_00007g2e_xyz-enrich.cif.gz Display(219.97 KB)
pdb_00007g2e_xyz-enrich.cif
no-atompdb_00007g2e_xyz-no-atom-enrich.xml.gz Display(61.89 KB)
pdb_00007g2e_xyz-no-atom-enrich.xml
ng-only7g2e-plus.json.gz Display(4.71 KB)
7g2e-plus.json
PDBpdb7g2e.ent.gz Display(153.32 KB)
pdb7g2e.ent
RDF7g2e.rdf.gz Visualize(146.86 KB)
7g2e.rdf
Structure factorsr7g2esf.ent.gz Display(12.01 MB)
r7g2esf.ent
Biological unit (mmCIF format)7g2e-assembly1.cif.gz Display(186.16 KB)
7g2e-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)7g2e.pdb1.gz Display(146.21 KB)
7g2e.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF7g2e_validation.pdf.gz Display(1.09 MB)
7g2e_validation.pdf
PDF-full7g2e_full_validation.pdf.gz Display(1.10 MB)
7g2e_full_validation.pdf
mmCIF7g2e_validation.cif.gz Display(56.32 KB)
7g2e_validation.cif
XML7g2e_validation.xml.gz Display(39.72 KB)
7g2e_validation.xml
PNG7g2e_multipercentile_validation.png.gz Display(163.72 KB)
7g2e_multipercentile_validation.png
SVG7g2e_multipercentile_validation.svg.gz Display(953.00 B)
7g2e_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)7g2e_validation_2fo-fc_map_coef.cif.gz Display(1.36 MB)
7g2e_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)7g2e_validation_fo-fc_map_coef.cif.gz Display(1.36 MB)
7g2e_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)7g2e_validation_2fo-fc_map_coef.mtz Visualize(2.23 MB)
fo-fc (MTZ)7g2e_validation_fo-fc_map_coef.mtz Visualize(2.23 MB)

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PDB entries from 2025-06-18

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