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6XIH

Structure-guided optimization of a novel class of ASK1 inhibitors with increased sp3 character and an exquisite selectivity profile

Resources
File formatFile name (file size)
PDBx/mmCIF6xih.cif.gz Display(220.18 KB)
6xih.cif
PDBx/mmJSONall6xih.json.gz Display (Tree)(148.91 KB)
6xih.json
no-atom6xih-noatom.json.gz Display (Header)(16.75 KB)
6xih-noatom.json
add only6xih-plus.json.gz Display(1.10 KB)
6xih-plus.json
PDBMLall6xih.xml.gz Display(297.09 KB)
6xih.xml
no-atom6xih-noatom.xml.gz Display(31.94 KB)
6xih-noatom.xml
ext-atom6xih-extatom.xml.gz Display(93.39 KB)
6xih-extatom.xml
PDBpdb6xih.ent.gz Display(176.84 KB)
pdb6xih.ent
RDF6xih.rdf.gz Visualize(92.19 KB)
6xih.rdf
Structure factorsr6xihsf.ent.gz Display(689.12 KB)
r6xihsf.ent
Biological unit (mmCIF format)6xih-assembly1.cif.gz Display(110.93 KB)
6xih-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

6xih-assembly2.cif.gz Display(105.74 KB)
6xih-assembly2.cif (B)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)6xih.pdb1.gz Display(88.53 KB)
6xih.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

6xih.pdb2.gz Display(85.27 KB)
6xih.pdb2 (B)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF6xih_validation.pdf.gz Display(998.36 KB)
6xih_validation.pdf
PDF-full6xih_full_validation.pdf.gz Display(1004.10 KB)
6xih_full_validation.pdf
mmCIF6xih_validation.cif.gz Display(27.34 KB)
6xih_validation.cif
XML6xih_validation.xml.gz Display(20.31 KB)
6xih_validation.xml
PNG6xih_multipercentile_validation.png.gz Display(169.63 KB)
6xih_multipercentile_validation.png
SVG6xih_multipercentile_validation.svg.gz Display(957.00 B)
6xih_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)6xih_validation_2fo-fc_map_coef.cif.gz Display(238.26 KB)
6xih_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)6xih_validation_fo-fc_map_coef.cif.gz Display(234.59 KB)
6xih_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)6xih_validation_2fo-fc_map_coef.mtz Visualize(574.48 KB)
fo-fc (MTZ)6xih_validation_fo-fc_map_coef.mtz Visualize(574.48 KB)

222415

PDB entries from 2024-07-10

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