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6UCS

Discovery and Structure-Based optimization of potent and selective WDR5 inhibitors containing a dihydroisoquinolinone bicyclic core

Resources
File formatFile name (file size)
PDBx/mmCIF6ucs.cif.gz Display(253.91 KB)
6ucs.cif
PDBx/mmJSONall6ucs.json.gz Display (Tree)(170.96 KB)
6ucs.json
no-atom6ucs-noatom.json.gz Display (Header)(19.48 KB)
6ucs-noatom.json
add only6ucs-plus.json.gz Display(1.73 KB)
6ucs-plus.json
PDBMLall6ucs.xml.gz Display(351.03 KB)
6ucs.xml
no-atom6ucs-noatom.xml.gz Display(38.82 KB)
6ucs-noatom.xml
ext-atom6ucs-extatom.xml.gz Display(116.36 KB)
6ucs-extatom.xml
PDBpdb6ucs.ent.gz Display(202.29 KB)
pdb6ucs.ent
RDF6ucs.rdf.gz Visualize(108.24 KB)
6ucs.rdf
Structure factorsr6ucssf.ent.gz Display(1.12 MB)
r6ucssf.ent
Biological unit (mmCIF format)6ucs-assembly1.cif.gz Display(126.46 KB)
6ucs-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

6ucs-assembly2.cif.gz Display(124.19 KB)
6ucs-assembly2.cif (B)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)6ucs.pdb1.gz Display(100.60 KB)
6ucs.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

6ucs.pdb2.gz Display(99.01 KB)
6ucs.pdb2 (B)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF6ucs_validation.pdf.gz Display(1.01 MB)
6ucs_validation.pdf
PDF-full6ucs_full_validation.pdf.gz Display(1.01 MB)
6ucs_full_validation.pdf
mmCIF6ucs_validation.cif.gz Display(41.14 KB)
6ucs_validation.cif
XML6ucs_validation.xml.gz Display(28.04 KB)
6ucs_validation.xml
PNG6ucs_multipercentile_validation.png.gz Display(164.03 KB)
6ucs_multipercentile_validation.png
SVG6ucs_multipercentile_validation.svg.gz Display(953.00 B)
6ucs_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)6ucs_validation_2fo-fc_map_coef.cif.gz Display(476.73 KB)
6ucs_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)6ucs_validation_fo-fc_map_coef.cif.gz Display(442.43 KB)
6ucs_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)6ucs_validation_2fo-fc_map_coef.mtz Visualize(1.10 MB)
fo-fc (MTZ)6ucs_validation_fo-fc_map_coef.mtz Visualize(1.10 MB)

219140

PDB entries from 2024-05-01

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