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6TPE

Fragment-based discovery of pyrazolopyridones as JAK1 inhibitors with excellent subtype selectivity

Resources
File formatFile name (file size)
PDBx/mmCIF6tpe.cif.gz Display(248.44 KB)
6tpe.cif
PDBx/mmJSONall6tpe.json.gz Display (Tree)(166.45 KB)
6tpe.json
no-atom6tpe-noatom.json.gz Display (Header)(17.13 KB)
6tpe-noatom.json
add only6tpe-plus.json.gz Display(1.14 KB)
6tpe-plus.json
PDBMLall6tpe.xml.gz Display(337.71 KB)
6tpe.xml
no-atom6tpe-noatom.xml.gz Display(35.38 KB)
6tpe-noatom.xml
ext-atom6tpe-extatom.xml.gz Display(105.52 KB)
6tpe-extatom.xml
pdb_nextgenallpdb_00006tpe_xyz-enrich.cif.gz Display(263.00 KB)
pdb_00006tpe_xyz-enrich.cif
no-atompdb_00006tpe_xyz-no-atom-enrich.xml.gz Display(50.00 KB)
pdb_00006tpe_xyz-no-atom-enrich.xml
ng-only6tpe-plus.json.gz Display(3.08 KB)
6tpe-plus.json
PDBpdb6tpe.ent.gz Display(200.94 KB)
pdb6tpe.ent
RDF6tpe.rdf.gz Visualize(101.31 KB)
6tpe.rdf
Structure factorsr6tpesf.ent.gz Display(286.86 KB)
r6tpesf.ent
Biological unit (mmCIF format)6tpe-assembly1.cif.gz Display(121.73 KB)
6tpe-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

6tpe-assembly2.cif.gz Display(122.61 KB)
6tpe-assembly2.cif (B)

*author defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)6tpe.pdb1.gz Display(98.13 KB)
6tpe.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

6tpe.pdb2.gz Display(99.15 KB)
6tpe.pdb2 (B)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF6tpe_validation.pdf.gz Display(801.94 KB)
6tpe_validation.pdf
PDF-full6tpe_full_validation.pdf.gz Display(802.52 KB)
6tpe_full_validation.pdf
mmCIF6tpe_validation.cif.gz Display(28.86 KB)
6tpe_validation.cif
XML6tpe_validation.xml.gz Display(22.86 KB)
6tpe_validation.xml
PNG6tpe_multipercentile_validation.png.gz Display(160.70 KB)
6tpe_multipercentile_validation.png
SVG6tpe_multipercentile_validation.svg.gz Display(904.00 B)
6tpe_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)6tpe_validation_2fo-fc_map_coef.cif.gz Display(224.05 KB)
6tpe_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)6tpe_validation_fo-fc_map_coef.cif.gz Display(223.60 KB)
6tpe_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)6tpe_validation_2fo-fc_map_coef.mtz Visualize(348.84 KB)
fo-fc (MTZ)6tpe_validation_fo-fc_map_coef.mtz Visualize(348.84 KB)

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PDB entries from 2025-06-11

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