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6TPD

Fragment-based discovery of pyrazolopyridones as JAK1 inhibitors with excellent subtype selectivity

Resources
File formatFile name (file size)
PDBx/mmCIF6tpd.cif.gz Display(134.61 KB)
6tpd.cif
PDBx/mmJSONall6tpd.json.gz Display (Tree)(95.52 KB)
6tpd.json
no-atom6tpd-noatom.json.gz Display (Header)(14.83 KB)
6tpd-noatom.json
add only6tpd-plus.json.gz Display(1.14 KB)
6tpd-plus.json
PDBMLall6tpd.xml.gz Display(180.30 KB)
6tpd.xml
no-atom6tpd-noatom.xml.gz Display(24.45 KB)
6tpd-noatom.xml
ext-atom6tpd-extatom.xml.gz Display(57.14 KB)
6tpd-extatom.xml
pdb_nextgenallpdb_00006tpd_xyz-enrich.cif.gz Display(142.33 KB)
pdb_00006tpd_xyz-enrich.cif
no-atompdb_00006tpd_xyz-no-atom-enrich.xml.gz Display(32.35 KB)
pdb_00006tpd_xyz-no-atom-enrich.xml
ng-only6tpd-plus.json.gz Display(2.59 KB)
6tpd-plus.json
PDBpdb6tpd.ent.gz Display(103.88 KB)
pdb6tpd.ent
RDF6tpd.rdf.gz Visualize(71.54 KB)
6tpd.rdf
Structure factorsr6tpdsf.ent.gz Display(738.80 KB)
r6tpdsf.ent
Biological unit (mmCIF format)6tpd-assembly1.cif.gz Display(125.13 KB)
6tpd-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)6tpd.pdb1.gz Display(98.91 KB)
6tpd.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF6tpd_validation.pdf.gz Display(769.67 KB)
6tpd_validation.pdf
PDF-full6tpd_full_validation.pdf.gz Display(772.79 KB)
6tpd_full_validation.pdf
mmCIF6tpd_validation.cif.gz Display(19.23 KB)
6tpd_validation.cif
XML6tpd_validation.xml.gz Display(13.96 KB)
6tpd_validation.xml
PNG6tpd_multipercentile_validation.png.gz Display(170.35 KB)
6tpd_multipercentile_validation.png
SVG6tpd_multipercentile_validation.svg.gz Display(976.00 B)
6tpd_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)6tpd_validation_2fo-fc_map_coef.cif.gz Display(382.68 KB)
6tpd_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)6tpd_validation_fo-fc_map_coef.cif.gz Display(379.46 KB)
6tpd_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)6tpd_validation_2fo-fc_map_coef.mtz Visualize(601.25 KB)
fo-fc (MTZ)6tpd_validation_fo-fc_map_coef.mtz Visualize(601.25 KB)

237735

PDB entries from 2025-06-18

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