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6P5M

Discovery of a Novel, Highly Potent, and Selective Thieno[3,2-d]pyrimidinone-Based Cdc7 inhibitor with a Quinuclidine Moiety (TAK-931) as an Orally Active Investigational Anti-Tumor Agent

Resources
File formatFile name (file size)
PDBx/mmCIF6p5m.cif.gz Display(635.34 KB)
6p5m.cif
PDBx/mmJSONall6p5m.json.gz Display (Tree)(412.46 KB)
6p5m.json
no-atom6p5m-noatom.json.gz Display (Header)(20.43 KB)
6p5m-noatom.json
add only6p5m-plus.json.gz Display(1.11 KB)
6p5m-plus.json
PDBMLall6p5m.xml.gz Display(880.02 KB)
6p5m.xml
no-atom6p5m-noatom.xml.gz Display(52.95 KB)
6p5m-noatom.xml
ext-atom6p5m-extatom.xml.gz Display(289.29 KB)
6p5m-extatom.xml
PDBpdb6p5m.ent.gz Display(531.37 KB)
pdb6p5m.ent
RDF6p5m.rdf.gz Visualize(153.58 KB)
6p5m.rdf
Structure factorsr6p5msf.ent.gz Display(2.36 MB)
r6p5msf.ent
Biological unit (mmCIF format)6p5m-assembly1.cif.gz Display(166.31 KB)
6p5m-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

6p5m-assembly2.cif.gz Display(162.54 KB)
6p5m-assembly2.cif (B)

*author defined assembly, 1 molecule(s) (monomeric)

6p5m-assembly3.cif.gz Display(163.69 KB)
6p5m-assembly3.cif (C)

*author defined assembly, 1 molecule(s) (monomeric)

6p5m-assembly4.cif.gz Display(163.11 KB)
6p5m-assembly4.cif (D)

*author defined assembly, 1 molecule(s) (monomeric)

6p5m-assembly5.cif.gz Display(320.78 KB)
6p5m-assembly5.cif (A,D)

*software defined assembly, 2 molecule(s) (dimeric)

6p5m-assembly6.cif.gz Display(317.95 KB)
6p5m-assembly6.cif (B,C)

*software defined assembly, 2 molecule(s) (dimeric)

Biological unit (PDB format)6p5m.pdb1.gz Display(137.06 KB)
6p5m.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

6p5m.pdb2.gz Display(132.77 KB)
6p5m.pdb2 (B)

*author defined assembly, 1 molecule(s) (monomeric)

6p5m.pdb3.gz Display(134.63 KB)
6p5m.pdb3 (C)

*author defined assembly, 1 molecule(s) (monomeric)

6p5m.pdb4.gz Display(133.63 KB)
6p5m.pdb4 (D)

*author defined assembly, 1 molecule(s) (monomeric)

6p5m.pdb5.gz Display(266.12 KB)
6p5m.pdb5 (A,D)

*software defined assembly, 2 molecule(s) (dimeric)

6p5m.pdb6.gz Display(262.86 KB)
6p5m.pdb6 (B,C)

*software defined assembly, 2 molecule(s) (dimeric)

Validation reportsPDF6p5m_validation.pdf.gz Display(989.35 KB)
6p5m_validation.pdf
PDF-full6p5m_full_validation.pdf.gz Display(1006.47 KB)
6p5m_full_validation.pdf
mmCIF6p5m_validation.cif.gz Display(72.43 KB)
6p5m_validation.cif
XML6p5m_validation.xml.gz Display(53.87 KB)
6p5m_validation.xml
PNG6p5m_multipercentile_validation.png.gz Display(167.21 KB)
6p5m_multipercentile_validation.png
SVG6p5m_multipercentile_validation.svg.gz Display(973.00 B)
6p5m_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)6p5m_validation_2fo-fc_map_coef.cif.gz Display(841.32 KB)
6p5m_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)6p5m_validation_fo-fc_map_coef.cif.gz Display(821.02 KB)
6p5m_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)6p5m_validation_2fo-fc_map_coef.mtz Visualize(1.91 MB)
fo-fc (MTZ)6p5m_validation_fo-fc_map_coef.mtz Visualize(1.91 MB)

219140

PDB entries from 2024-05-01

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