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6GDM

Fragment-based discovery of a highly potent, orally bioavailable inhibitor which modulates the phosphorylation and catalytic activity of ERK1/2

Resources
File formatFile name (file size)
PDBx/mmCIF6gdm.cif.gz Display(166.19 KB)
6gdm.cif
PDBx/mmJSONall6gdm.json.gz Display (Tree)(119.45 KB)
6gdm.json
no-atom6gdm-noatom.json.gz Display (Header)(16.53 KB)
6gdm-noatom.json
add only6gdm-plus.json.gz Display(2.94 KB)
6gdm-plus.json
PDBMLall6gdm.xml.gz Display(223.15 KB)
6gdm.xml
no-atom6gdm-noatom.xml.gz Display(25.22 KB)
6gdm-noatom.xml
ext-atom6gdm-extatom.xml.gz Display(75.19 KB)
6gdm-extatom.xml
PDBpdb6gdm.ent.gz Display(135.43 KB)
pdb6gdm.ent
RDF6gdm.rdf.gz Visualize(60.16 KB)
6gdm.rdf
Structure factorsr6gdmsf.ent.gz Display(552.37 KB)
r6gdmsf.ent
Biological unit (mmCIF format)6gdm-assembly1.cif.gz Display(159.58 KB)
6gdm-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)6gdm.pdb1.gz Display(129.32 KB)
6gdm.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF6gdm_validation.pdf.gz Display(691.23 KB)
6gdm_validation.pdf
PDF-full6gdm_full_validation.pdf.gz Display(694.31 KB)
6gdm_full_validation.pdf
mmCIF6gdm_validation.cif.gz Display(29.44 KB)
6gdm_validation.cif
XML6gdm_validation.xml.gz Display(19.24 KB)
6gdm_validation.xml
PNG6gdm_multipercentile_validation.png.gz Display(167.11 KB)
6gdm_multipercentile_validation.png
SVG6gdm_multipercentile_validation.svg.gz Display(957.00 B)
6gdm_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)6gdm_validation_2fo-fc_map_coef.cif.gz Display(444.69 KB)
6gdm_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)6gdm_validation_fo-fc_map_coef.cif.gz Display(440.63 KB)
6gdm_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)6gdm_validation_2fo-fc_map_coef.mtz Visualize(713.52 KB)
fo-fc (MTZ)6gdm_validation_fo-fc_map_coef.mtz Visualize(713.52 KB)

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PDB entries from 2024-07-10

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