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6G9M

Fragment-based discovery of a highly potent, orally bioavailable inhibitor which modulates the phosphorylation and catalytic activity of ERK1/2

Resources
File formatFile name (file size)
PDBx/mmCIF6g9m.cif.gz Display(166.28 KB)
6g9m.cif
PDBx/mmJSONall6g9m.json.gz Display (Tree)(119.53 KB)
6g9m.json
no-atom6g9m-noatom.json.gz Display (Header)(17.00 KB)
6g9m-noatom.json
add only6g9m-plus.json.gz Display(2.93 KB)
6g9m-plus.json
PDBMLall6g9m.xml.gz Display(223.21 KB)
6g9m.xml
no-atom6g9m-noatom.xml.gz Display(25.65 KB)
6g9m-noatom.xml
ext-atom6g9m-extatom.xml.gz Display(75.98 KB)
6g9m-extatom.xml
PDBpdb6g9m.ent.gz Display(134.50 KB)
pdb6g9m.ent
RDF6g9m.rdf.gz Visualize(61.25 KB)
6g9m.rdf
Structure factorsr6g9msf.ent.gz Display(501.82 KB)
r6g9msf.ent
Biological unit (mmCIF format)6g9m-assembly1.cif.gz Display(159.87 KB)
6g9m-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)6g9m.pdb1.gz Display(129.23 KB)
6g9m.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF6g9m_validation.pdf.gz Display(594.78 KB)
6g9m_validation.pdf
PDF-full6g9m_full_validation.pdf.gz Display(596.21 KB)
6g9m_full_validation.pdf
XML6g9m_validation.xml.gz Display(20.37 KB)
6g9m_validation.xml
PNG6g9m_multipercentile_validation.png.gz Display(144.51 KB)
6g9m_multipercentile_validation.png
SVG6g9m_multipercentile_validation.svg.gz Display(944.00 B)
6g9m_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)6g9m_validation_2fo-fc_map_coef.cif.gz Display(320.45 KB)
6g9m_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)6g9m_validation_fo-fc_map_coef.cif.gz Display(306.00 KB)
6g9m_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)6g9m_validation_2fo-fc_map_coef.mtz Visualize(766.26 KB)
fo-fc (MTZ)6g9m_validation_fo-fc_map_coef.mtz Visualize(766.26 KB)

221051

PDB entries from 2024-06-12

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