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6G9K

Fragment-based discovery of a highly potent, orally bioavailable inhibitor which modulates the phosphorylation and catalytic activity of ERK1/2

Resources
File formatFile name (file size)
PDBx/mmCIF6g9k.cif.gz Display(165.14 KB)
6g9k.cif
PDBx/mmJSONall6g9k.json.gz Display (Tree)(118.23 KB)
6g9k.json
no-atom6g9k-noatom.json.gz Display (Header)(16.42 KB)
6g9k-noatom.json
add only6g9k-plus.json.gz Display(2.94 KB)
6g9k-plus.json
PDBMLall6g9k.xml.gz Display(221.60 KB)
6g9k.xml
no-atom6g9k-noatom.xml.gz Display(24.87 KB)
6g9k-noatom.xml
ext-atom6g9k-extatom.xml.gz Display(74.94 KB)
6g9k-extatom.xml
PDBpdb6g9k.ent.gz Display(133.82 KB)
pdb6g9k.ent
RDF6g9k.rdf.gz Visualize(59.93 KB)
6g9k.rdf
Structure factorsr6g9ksf.ent.gz Display(449.58 KB)
r6g9ksf.ent
Biological unit (mmCIF format)6g9k-assembly1.cif.gz Display(158.54 KB)
6g9k-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)6g9k.pdb1.gz Display(128.60 KB)
6g9k.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF6g9k_validation.pdf.gz Display(702.60 KB)
6g9k_validation.pdf
PDF-full6g9k_full_validation.pdf.gz Display(703.01 KB)
6g9k_full_validation.pdf
mmCIF6g9k_validation.cif.gz Display(29.17 KB)
6g9k_validation.cif
XML6g9k_validation.xml.gz Display(18.72 KB)
6g9k_validation.xml
PNG6g9k_multipercentile_validation.png.gz Display(168.34 KB)
6g9k_multipercentile_validation.png
SVG6g9k_multipercentile_validation.svg.gz Display(972.00 B)
6g9k_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)6g9k_validation_2fo-fc_map_coef.cif.gz Display(414.37 KB)
6g9k_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)6g9k_validation_fo-fc_map_coef.cif.gz Display(415.07 KB)
6g9k_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)6g9k_validation_2fo-fc_map_coef.mtz Visualize(665.69 KB)
fo-fc (MTZ)6g9k_validation_fo-fc_map_coef.mtz Visualize(665.69 KB)

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PDB entries from 2024-07-17

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