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6G9H

Fragment-based discovery of a highly potent, orally bioavailable inhibitor which modulates the phosphorylation and catalytic activity of ERK1/2

Resources
File formatFile name (file size)
PDBx/mmCIF6g9h.cif.gz Display(165.39 KB)
6g9h.cif
PDBx/mmJSONall6g9h.json.gz Display (Tree)(118.44 KB)
6g9h.json
no-atom6g9h-noatom.json.gz Display (Header)(16.81 KB)
6g9h-noatom.json
add only6g9h-plus.json.gz Display(2.94 KB)
6g9h-plus.json
PDBMLall6g9h.xml.gz Display(222.02 KB)
6g9h.xml
no-atom6g9h-noatom.xml.gz Display(25.55 KB)
6g9h-noatom.xml
ext-atom6g9h-extatom.xml.gz Display(75.80 KB)
6g9h-extatom.xml
PDBpdb6g9h.ent.gz Display(133.59 KB)
pdb6g9h.ent
RDF6g9h.rdf.gz Visualize(61.00 KB)
6g9h.rdf
Structure factorsr6g9hsf.ent.gz Display(617.48 KB)
r6g9hsf.ent
Biological unit (mmCIF format)6g9h-assembly1.cif.gz Display(158.64 KB)
6g9h-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)6g9h.pdb1.gz Display(128.45 KB)
6g9h.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF6g9h_validation.pdf.gz Display(755.10 KB)
6g9h_validation.pdf
PDF-full6g9h_full_validation.pdf.gz Display(757.35 KB)
6g9h_full_validation.pdf
mmCIF6g9h_validation.cif.gz Display(30.15 KB)
6g9h_validation.cif
XML6g9h_validation.xml.gz Display(19.19 KB)
6g9h_validation.xml
PNG6g9h_multipercentile_validation.png.gz Display(163.21 KB)
6g9h_multipercentile_validation.png
SVG6g9h_multipercentile_validation.svg.gz Display(949.00 B)
6g9h_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)6g9h_validation_2fo-fc_map_coef.cif.gz Display(590.06 KB)
6g9h_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)6g9h_validation_fo-fc_map_coef.cif.gz Display(562.43 KB)
6g9h_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)6g9h_validation_2fo-fc_map_coef.mtz Visualize(955.84 KB)
fo-fc (MTZ)6g9h_validation_fo-fc_map_coef.mtz Visualize(955.84 KB)

222415

PDB entries from 2024-07-10

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