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6G9A

Fragment-based discovery of a highly potent, orally bioavailable inhibitor which modulates the phosphorylation and catalytic activity of ERK1/2

Resources
File formatFile name (file size)
PDBx/mmCIF6g9a.cif.gz Display(166.70 KB)
6g9a.cif
PDBx/mmJSONall6g9a.json.gz Display (Tree)(119.81 KB)
6g9a.json
no-atom6g9a-noatom.json.gz Display (Header)(17.06 KB)
6g9a-noatom.json
add only6g9a-plus.json.gz Display(2.93 KB)
6g9a-plus.json
PDBMLall6g9a.xml.gz Display(223.38 KB)
6g9a.xml
no-atom6g9a-noatom.xml.gz Display(25.85 KB)
6g9a-noatom.xml
ext-atom6g9a-extatom.xml.gz Display(76.16 KB)
6g9a-extatom.xml
PDBpdb6g9a.ent.gz Display(134.42 KB)
pdb6g9a.ent
RDF6g9a.rdf.gz Visualize(61.46 KB)
6g9a.rdf
Structure factorsr6g9asf.ent.gz Display(460.42 KB)
r6g9asf.ent
Biological unit (mmCIF format)6g9a-assembly1.cif.gz Display(160.32 KB)
6g9a-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)6g9a.pdb1.gz Display(129.30 KB)
6g9a.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF6g9a_validation.pdf.gz Display(758.99 KB)
6g9a_validation.pdf
PDF-full6g9a_full_validation.pdf.gz Display(760.27 KB)
6g9a_full_validation.pdf
mmCIF6g9a_validation.cif.gz Display(31.07 KB)
6g9a_validation.cif
XML6g9a_validation.xml.gz Display(19.70 KB)
6g9a_validation.xml
PNG6g9a_multipercentile_validation.png.gz Display(165.86 KB)
6g9a_multipercentile_validation.png
SVG6g9a_multipercentile_validation.svg.gz Display(955.00 B)
6g9a_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)6g9a_validation_2fo-fc_map_coef.cif.gz Display(444.90 KB)
6g9a_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)6g9a_validation_fo-fc_map_coef.cif.gz Display(443.70 KB)
6g9a_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)6g9a_validation_2fo-fc_map_coef.mtz Visualize(708.48 KB)
fo-fc (MTZ)6g9a_validation_fo-fc_map_coef.mtz Visualize(708.48 KB)

223532

PDB entries from 2024-08-07

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