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6G8X

Fragment-based discovery of a highly potent, orally bioavailable inhibitor which modulates the phosphorylation and catalytic activity of ERK1/2

Resources
File formatFile name (file size)
PDBx/mmCIF6g8x.cif.gz Display(161.53 KB)
6g8x.cif
PDBx/mmJSONall6g8x.json.gz Display (Tree)(115.03 KB)
6g8x.json
no-atom6g8x-noatom.json.gz Display (Header)(16.35 KB)
6g8x-noatom.json
add only6g8x-plus.json.gz Display(2.94 KB)
6g8x-plus.json
PDBMLall6g8x.xml.gz Display(216.66 KB)
6g8x.xml
no-atom6g8x-noatom.xml.gz Display(24.72 KB)
6g8x-noatom.xml
ext-atom6g8x-extatom.xml.gz Display(73.53 KB)
6g8x-extatom.xml
PDBpdb6g8x.ent.gz Display(129.97 KB)
pdb6g8x.ent
RDF6g8x.rdf.gz Visualize(59.50 KB)
6g8x.rdf
Structure factorsr6g8xsf.ent.gz Display(648.93 KB)
r6g8xsf.ent
Biological unit (mmCIF format)6g8x-assembly1.cif.gz Display(155.04 KB)
6g8x-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)6g8x.pdb1.gz Display(125.08 KB)
6g8x.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF6g8x_validation.pdf.gz Display(1023.73 KB)
6g8x_validation.pdf
PDF-full6g8x_full_validation.pdf.gz Display(1.00 MB)
6g8x_full_validation.pdf
mmCIF6g8x_validation.cif.gz Display(29.11 KB)
6g8x_validation.cif
XML6g8x_validation.xml.gz Display(18.70 KB)
6g8x_validation.xml
PNG6g8x_multipercentile_validation.png.gz Display(172.64 KB)
6g8x_multipercentile_validation.png
SVG6g8x_multipercentile_validation.svg.gz Display(974.00 B)
6g8x_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)6g8x_validation_2fo-fc_map_coef.cif.gz Display(548.49 KB)
6g8x_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)6g8x_validation_fo-fc_map_coef.cif.gz Display(508.08 KB)
6g8x_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)6g8x_validation_2fo-fc_map_coef.mtz Visualize(907.91 KB)
fo-fc (MTZ)6g8x_validation_fo-fc_map_coef.mtz Visualize(907.91 KB)

222415

PDB entries from 2024-07-10

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