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6DAS

Discovery of Potent 2-Aryl-6,7-Dihydro-5HPyrrolo[ 1,2-a]imidazoles as WDR5 WIN-site Inhibitors Using Fragment-Based Methods and Structure-Based Design

Resources
File formatFile name (file size)
PDBx/mmCIF6das.cif.gz Display(260.56 KB)
6das.cif
PDBx/mmJSONall6das.json.gz Display (Tree)(175.07 KB)
6das.json
no-atom6das-noatom.json.gz Display (Header)(18.36 KB)
6das-noatom.json
add only6das-plus.json.gz Display(1.73 KB)
6das-plus.json
PDBMLall6das.xml.gz Display(363.74 KB)
6das.xml
no-atom6das-noatom.xml.gz Display(37.75 KB)
6das-noatom.xml
ext-atom6das-extatom.xml.gz Display(119.80 KB)
6das-extatom.xml
PDBpdb6das.ent.gz Display(207.96 KB)
pdb6das.ent
RDF6das.rdf.gz Visualize(105.41 KB)
6das.rdf
Structure factorsr6dassf.ent.gz Display(1.09 MB)
r6dassf.ent
Biological unit (mmCIF format)6das-assembly1.cif.gz Display(131.24 KB)
6das-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

6das-assembly2.cif.gz Display(128.90 KB)
6das-assembly2.cif (B)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)6das.pdb1.gz Display(104.53 KB)
6das.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

6das.pdb2.gz Display(101.53 KB)
6das.pdb2 (B)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF6das_validation.pdf.gz Display(1.02 MB)
6das_validation.pdf
PDF-full6das_full_validation.pdf.gz Display(1.02 MB)
6das_full_validation.pdf
mmCIF6das_validation.cif.gz Display(45.82 KB)
6das_validation.cif
XML6das_validation.xml.gz Display(30.07 KB)
6das_validation.xml
PNG6das_multipercentile_validation.png.gz Display(159.16 KB)
6das_multipercentile_validation.png
SVG6das_multipercentile_validation.svg.gz Display(949.00 B)
6das_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)6das_validation_2fo-fc_map_coef.cif.gz Display(534.44 KB)
6das_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)6das_validation_fo-fc_map_coef.cif.gz Display(509.16 KB)
6das_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)6das_validation_2fo-fc_map_coef.mtz Visualize(1.23 MB)
fo-fc (MTZ)6das_validation_fo-fc_map_coef.mtz Visualize(1.23 MB)

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PDB entries from 2024-07-17

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