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5UK8

The co-structure of (R)-4-(6-(1-(cyclopropylsulfonyl)cyclopropyl)-2-(1H-indol-4-yl)pyrimidin-4-yl)-3-methylmorpholine and a rationally designed PI3K-alpha mutant that mimics ATR

Resources
File formatFile name (file size)
PDBx/mmCIF5uk8.cif.gz Display(406.34 KB)
5uk8.cif
PDBx/mmJSONall5uk8.json.gz Display (Tree)(295.41 KB)
5uk8.json
no-atom5uk8-noatom.json.gz Display (Header)(29.35 KB)
5uk8-noatom.json
add only5uk8-plus.json.gz Display(2.43 KB)
5uk8-plus.json
PDBMLall5uk8.xml.gz Display(614.83 KB)
5uk8.xml
no-atom5uk8-noatom.xml.gz Display(57.69 KB)
5uk8-noatom.xml
ext-atom5uk8-extatom.xml.gz Display(234.72 KB)
5uk8-extatom.xml
PDBpdb5uk8.ent.gz Display(312.20 KB)
pdb5uk8.ent
RDF5uk8.rdf.gz Visualize(175.17 KB)
5uk8.rdf
Structure factorsr5uk8sf.ent.gz Display(2.16 MB)
r5uk8sf.ent
Biological unit (mmCIF format)5uk8-assembly1.cif.gz Display(395.50 KB)
5uk8-assembly1.cif (A,B)

*author and software defined assembly, 2 molecule(s) (dimeric)

Biological unit (PDB format)5uk8.pdb1.gz Display(305.47 KB)
5uk8.pdb1 (A,B)

*author and software defined assembly, 2 molecule(s) (dimeric)

Validation reportsPDF5uk8_validation.pdf.gz Display(850.40 KB)
5uk8_validation.pdf
PDF-full5uk8_full_validation.pdf.gz Display(857.86 KB)
5uk8_full_validation.pdf
mmCIF5uk8_validation.cif.gz Display(61.89 KB)
5uk8_validation.cif
XML5uk8_validation.xml.gz Display(44.02 KB)
5uk8_validation.xml
PNG5uk8_multipercentile_validation.png.gz Display(170.93 KB)
5uk8_multipercentile_validation.png
SVG5uk8_multipercentile_validation.svg.gz Display(978.00 B)
5uk8_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)5uk8_validation_2fo-fc_map_coef.cif.gz Display(777.98 KB)
5uk8_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)5uk8_validation_fo-fc_map_coef.cif.gz Display(775.24 KB)
5uk8_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)5uk8_validation_2fo-fc_map_coef.mtz Visualize(1.21 MB)
fo-fc (MTZ)5uk8_validation_fo-fc_map_coef.mtz Visualize(1.21 MB)

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PDB entries from 2024-07-24

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