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5UG9

Crystal structure of the EGFR kinase domain (L858R, T790M, V948R) in complex with a covalent inhibitor N-[(3R,4R)-4-fluoro-1-{6-[(3-methoxy-1-methyl-1H-pyrazol-4-yl)amino]-9-(propan-2-yl)-9H-purin-2-yl}pyrrolidin-3-yl]propanamide

Resources
File formatFile name (file size)
PDBx/mmCIF5ug9.cif.gz Display(79.71 KB)
5ug9.cif
PDBx/mmJSONall5ug9.json.gz Display (Tree)(58.31 KB)
5ug9.json
no-atom5ug9-noatom.json.gz Display (Header)(16.16 KB)
5ug9-noatom.json
add only5ug9-plus.json.gz Display(1.47 KB)
5ug9-plus.json
PDBMLall5ug9.xml.gz Display(102.61 KB)
5ug9.xml
no-atom5ug9-noatom.xml.gz Display(23.20 KB)
5ug9-noatom.xml
ext-atom5ug9-extatom.xml.gz Display(60.07 KB)
5ug9-extatom.xml
PDBpdb5ug9.ent.gz Display(60.61 KB)
pdb5ug9.ent
RDF5ug9.rdf.gz Visualize(55.97 KB)
5ug9.rdf
Structure factorsr5ug9sf.ent.gz Display(445.59 KB)
r5ug9sf.ent
Biological unit (mmCIF format)5ug9-assembly1.cif.gz Display(72.08 KB)
5ug9-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)5ug9.pdb1.gz Display(55.56 KB)
5ug9.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF5ug9_validation.pdf.gz Display(829.10 KB)
5ug9_validation.pdf
PDF-full5ug9_full_validation.pdf.gz Display(831.65 KB)
5ug9_full_validation.pdf
mmCIF5ug9_validation.cif.gz Display(23.90 KB)
5ug9_validation.cif
XML5ug9_validation.xml.gz Display(15.88 KB)
5ug9_validation.xml
PNG5ug9_multipercentile_validation.png.gz Display(167.54 KB)
5ug9_multipercentile_validation.png
SVG5ug9_multipercentile_validation.svg.gz Display(960.00 B)
5ug9_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)5ug9_validation_2fo-fc_map_coef.cif.gz Display(928.92 KB)
5ug9_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)5ug9_validation_fo-fc_map_coef.cif.gz Display(931.03 KB)
5ug9_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)5ug9_validation_2fo-fc_map_coef.mtz Visualize(1.47 MB)
fo-fc (MTZ)5ug9_validation_fo-fc_map_coef.mtz Visualize(1.47 MB)

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PDB entries from 2024-07-10

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