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5SKR

CRYSTAL STRUCTURE OF HUMAN PHOSPHODIESTERASE 10 IN COMPLEX WITH n1c(cc(n1C)NC(c2nn(cc2c3ccncc3)C)=O)c4ncccc4, micromolar IC50=0.124219

Resources
File formatFile name (file size)
PDBx/mmCIF5skr.cif.gz Display(278.39 KB)
5skr.cif
PDBx/mmJSONall5skr.json.gz Display (Tree)(171.54 KB)
5skr.json
no-atom5skr-noatom.json.gz Display (Header)(20.80 KB)
5skr-noatom.json
add only5skr-plus.json.gz Display(1009.00 B)
5skr-plus.json
PDBMLall5skr.xml.gz Display(380.01 KB)
5skr.xml
no-atom5skr-noatom.xml.gz Display(56.40 KB)
5skr-noatom.xml
ext-atom5skr-extatom.xml.gz Display(245.16 KB)
5skr-extatom.xml
pdb_nextgenallpdb_00005skr_xyz-enrich.cif.gz Display(304.20 KB)
pdb_00005skr_xyz-enrich.cif
no-atompdb_00005skr_xyz-no-atom-enrich.xml.gz Display(69.51 KB)
pdb_00005skr_xyz-no-atom-enrich.xml
ng-only5skr-plus.json.gz Display(3.42 KB)
5skr-plus.json
PDBpdb5skr.ent.gz Display(223.67 KB)
pdb5skr.ent
RDF5skr.rdf.gz Visualize(152.30 KB)
5skr.rdf
Structure factorsr5skrsf.ent.gz Display(14.30 MB)
r5skrsf.ent
Biological unit (mmCIF format)5skr-assembly1.cif.gz Display(72.49 KB)
5skr-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

5skr-assembly2.cif.gz Display(72.56 KB)
5skr-assembly2.cif (B)

*author defined assembly, 1 molecule(s) (monomeric)

5skr-assembly3.cif.gz Display(72.78 KB)
5skr-assembly3.cif (C)

*author defined assembly, 1 molecule(s) (monomeric)

5skr-assembly4.cif.gz Display(70.20 KB)
5skr-assembly4.cif (D)

*author defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)5skr.pdb1.gz Display(57.30 KB)
5skr.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

5skr.pdb2.gz Display(57.31 KB)
5skr.pdb2 (B)

*author defined assembly, 1 molecule(s) (monomeric)

5skr.pdb3.gz Display(57.65 KB)
5skr.pdb3 (C)

*author defined assembly, 1 molecule(s) (monomeric)

5skr.pdb4.gz Display(55.43 KB)
5skr.pdb4 (D)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF5skr_validation.pdf.gz Display(1.48 MB)
5skr_validation.pdf
PDF-full5skr_full_validation.pdf.gz Display(1.50 MB)
5skr_full_validation.pdf
mmCIF5skr_validation.cif.gz Display(79.28 KB)
5skr_validation.cif
XML5skr_validation.xml.gz Display(60.28 KB)
5skr_validation.xml
PNG5skr_multipercentile_validation.png.gz Display(169.34 KB)
5skr_multipercentile_validation.png
SVG5skr_multipercentile_validation.svg.gz Display(976.00 B)
5skr_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)5skr_validation_2fo-fc_map_coef.cif.gz Display(1.62 MB)
5skr_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)5skr_validation_fo-fc_map_coef.cif.gz Display(1.61 MB)
5skr_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)5skr_validation_2fo-fc_map_coef.mtz Visualize(2.53 MB)
fo-fc (MTZ)5skr_validation_fo-fc_map_coef.mtz Visualize(2.53 MB)

240971

PDB entries from 2025-08-27

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