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5SKL

CRYSTAL STRUCTURE OF HUMAN PHOSPHODIESTERASE 10 IN COMPLEX WITH c4(c(C(=O)Nc2cc1nc(cn1cc2C#N)c3ccccc3)n(C)nc4)C(=O)N5CCOCC5, micromolar IC50=0.000990

Resources
File formatFile name (file size)
PDBx/mmCIF5skl.cif.gz Display(273.87 KB)
5skl.cif
PDBx/mmJSONall5skl.json.gz Display (Tree)(168.83 KB)
5skl.json
no-atom5skl-noatom.json.gz Display (Header)(20.02 KB)
5skl-noatom.json
add only5skl-plus.json.gz Display(1016.00 B)
5skl-plus.json
PDBMLall5skl.xml.gz Display(374.49 KB)
5skl.xml
no-atom5skl-noatom.xml.gz Display(54.80 KB)
5skl-noatom.xml
ext-atom5skl-extatom.xml.gz Display(242.01 KB)
5skl-extatom.xml
pdb_nextgenallpdb_00005skl_xyz-enrich.cif.gz Display(299.28 KB)
pdb_00005skl_xyz-enrich.cif
no-atompdb_00005skl_xyz-no-atom-enrich.xml.gz Display(67.85 KB)
pdb_00005skl_xyz-no-atom-enrich.xml
ng-only5skl-plus.json.gz Display(3.42 KB)
5skl-plus.json
PDBpdb5skl.ent.gz Display(220.96 KB)
pdb5skl.ent
RDF5skl.rdf.gz Visualize(149.48 KB)
5skl.rdf
Structure factorsr5sklsf.ent.gz Display(8.73 MB)
r5sklsf.ent
Biological unit (mmCIF format)5skl-assembly1.cif.gz Display(71.43 KB)
5skl-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

5skl-assembly2.cif.gz Display(71.51 KB)
5skl-assembly2.cif (B)

*author defined assembly, 1 molecule(s) (monomeric)

5skl-assembly3.cif.gz Display(71.83 KB)
5skl-assembly3.cif (C)

*author defined assembly, 1 molecule(s) (monomeric)

5skl-assembly4.cif.gz Display(68.76 KB)
5skl-assembly4.cif (D)

*author defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)5skl.pdb1.gz Display(56.67 KB)
5skl.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

5skl.pdb2.gz Display(56.73 KB)
5skl.pdb2 (B)

*author defined assembly, 1 molecule(s) (monomeric)

5skl.pdb3.gz Display(56.87 KB)
5skl.pdb3 (C)

*author defined assembly, 1 molecule(s) (monomeric)

5skl.pdb4.gz Display(54.69 KB)
5skl.pdb4 (D)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF5skl_validation.pdf.gz Display(1.34 MB)
5skl_validation.pdf
PDF-full5skl_full_validation.pdf.gz Display(1.36 MB)
5skl_full_validation.pdf
mmCIF5skl_validation.cif.gz Display(75.05 KB)
5skl_validation.cif
XML5skl_validation.xml.gz Display(58.04 KB)
5skl_validation.xml
PNG5skl_multipercentile_validation.png.gz Display(167.23 KB)
5skl_multipercentile_validation.png
SVG5skl_multipercentile_validation.svg.gz Display(974.00 B)
5skl_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)5skl_validation_2fo-fc_map_coef.cif.gz Display(1.17 MB)
5skl_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)5skl_validation_fo-fc_map_coef.cif.gz Display(1.18 MB)
5skl_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)5skl_validation_2fo-fc_map_coef.mtz Visualize(1.85 MB)
fo-fc (MTZ)5skl_validation_fo-fc_map_coef.mtz Visualize(1.85 MB)

240971

PDB entries from 2025-08-27

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