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5SKF

CRYSTAL STRUCTURE OF HUMAN PHOSPHODIESTERASE 10 IN COMPLEX WITH C1(=NN(C=CC1=O)c2cccc3c2OC(O3)(F)F)c4ccnn4c5cccc(c5)C#N, micromolar IC50=0.080428

Resources
File formatFile name (file size)
PDBx/mmCIF5skf.cif.gz Display(279.12 KB)
5skf.cif
PDBx/mmJSONall5skf.json.gz Display (Tree)(173.51 KB)
5skf.json
no-atom5skf-noatom.json.gz Display (Header)(22.72 KB)
5skf-noatom.json
add only5skf-plus.json.gz Display(1.04 KB)
5skf-plus.json
PDBMLall5skf.xml.gz Display(381.67 KB)
5skf.xml
no-atom5skf-noatom.xml.gz Display(59.46 KB)
5skf-noatom.xml
ext-atom5skf-extatom.xml.gz Display(243.94 KB)
5skf-extatom.xml
pdb_nextgenallpdb_00005skf_xyz-enrich.cif.gz Display(304.71 KB)
pdb_00005skf_xyz-enrich.cif
no-atompdb_00005skf_xyz-no-atom-enrich.xml.gz Display(72.22 KB)
pdb_00005skf_xyz-no-atom-enrich.xml
ng-only5skf-plus.json.gz Display(3.41 KB)
5skf-plus.json
PDBpdb5skf.ent.gz Display(224.09 KB)
pdb5skf.ent
RDF5skf.rdf.gz Visualize(158.38 KB)
5skf.rdf
Structure factorsr5skfsf.ent.gz Display(10.38 MB)
r5skfsf.ent
Biological unit (mmCIF format)5skf-assembly1.cif.gz Display(71.91 KB)
5skf-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

5skf-assembly2.cif.gz Display(72.50 KB)
5skf-assembly2.cif (B)

*author defined assembly, 1 molecule(s) (monomeric)

5skf-assembly3.cif.gz Display(70.99 KB)
5skf-assembly3.cif (C)

*author defined assembly, 1 molecule(s) (monomeric)

5skf-assembly4.cif.gz Display(70.33 KB)
5skf-assembly4.cif (D)

*author defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)5skf.pdb1.gz Display(57.49 KB)
5skf.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

5skf.pdb2.gz Display(57.43 KB)
5skf.pdb2 (B)

*author defined assembly, 1 molecule(s) (monomeric)

5skf.pdb3.gz Display(57.07 KB)
5skf.pdb3 (C)

*author defined assembly, 1 molecule(s) (monomeric)

5skf.pdb4.gz Display(56.44 KB)
5skf.pdb4 (D)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF5skf_validation.pdf.gz Display(1.79 MB)
5skf_validation.pdf
PDF-full5skf_full_validation.pdf.gz Display(1.80 MB)
5skf_full_validation.pdf
mmCIF5skf_validation.cif.gz Display(75.79 KB)
5skf_validation.cif
XML5skf_validation.xml.gz Display(57.81 KB)
5skf_validation.xml
PNG5skf_multipercentile_validation.png.gz Display(163.35 KB)
5skf_multipercentile_validation.png
SVG5skf_multipercentile_validation.svg.gz Display(928.00 B)
5skf_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)5skf_validation_2fo-fc_map_coef.cif.gz Display(1.40 MB)
5skf_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)5skf_validation_fo-fc_map_coef.cif.gz Display(1.40 MB)
5skf_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)5skf_validation_2fo-fc_map_coef.mtz Visualize(2.13 MB)
fo-fc (MTZ)5skf_validation_fo-fc_map_coef.mtz Visualize(2.13 MB)

239149

PDB entries from 2025-07-23

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