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5SKE

CRYSTAL STRUCTURE OF HUMAN PHOSPHODIESTERASE 10 IN COMPLEX WITH c1nc(nc(c1Nc2cncnc2)C(Nc3cc(ccc3)OC(F)(F)F)=O)C(C)(C)C, micromolar IC50=0.037955

Resources
File formatFile name (file size)
PDBx/mmCIF5ske.cif.gz Display(273.67 KB)
5ske.cif
PDBx/mmJSONall5ske.json.gz Display (Tree)(168.64 KB)
5ske.json
no-atom5ske-noatom.json.gz Display (Header)(20.11 KB)
5ske-noatom.json
add only5ske-plus.json.gz Display(1015.00 B)
5ske-plus.json
PDBMLall5ske.xml.gz Display(374.02 KB)
5ske.xml
no-atom5ske-noatom.xml.gz Display(55.10 KB)
5ske-noatom.xml
ext-atom5ske-extatom.xml.gz Display(241.92 KB)
5ske-extatom.xml
pdb_nextgenallpdb_00005ske_xyz-enrich.cif.gz Display(299.03 KB)
pdb_00005ske_xyz-enrich.cif
no-atompdb_00005ske_xyz-no-atom-enrich.xml.gz Display(68.15 KB)
pdb_00005ske_xyz-no-atom-enrich.xml
ng-only5ske-plus.json.gz Display(3.42 KB)
5ske-plus.json
PDBpdb5ske.ent.gz Display(220.65 KB)
pdb5ske.ent
RDF5ske.rdf.gz Visualize(149.86 KB)
5ske.rdf
Structure factorsr5skesf.ent.gz Display(10.55 MB)
r5skesf.ent
Biological unit (mmCIF format)5ske-assembly1.cif.gz Display(71.15 KB)
5ske-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

5ske-assembly2.cif.gz Display(71.44 KB)
5ske-assembly2.cif (B)

*author defined assembly, 1 molecule(s) (monomeric)

5ske-assembly3.cif.gz Display(71.59 KB)
5ske-assembly3.cif (C)

*author defined assembly, 1 molecule(s) (monomeric)

5ske-assembly4.cif.gz Display(68.78 KB)
5ske-assembly4.cif (D)

*author defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)5ske.pdb1.gz Display(56.46 KB)
5ske.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

5ske.pdb2.gz Display(56.74 KB)
5ske.pdb2 (B)

*author defined assembly, 1 molecule(s) (monomeric)

5ske.pdb3.gz Display(56.82 KB)
5ske.pdb3 (C)

*author defined assembly, 1 molecule(s) (monomeric)

5ske.pdb4.gz Display(54.72 KB)
5ske.pdb4 (D)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF5ske_validation.pdf.gz Display(1.52 MB)
5ske_validation.pdf
PDF-full5ske_full_validation.pdf.gz Display(1.53 MB)
5ske_full_validation.pdf
mmCIF5ske_validation.cif.gz Display(71.09 KB)
5ske_validation.cif
XML5ske_validation.xml.gz Display(53.68 KB)
5ske_validation.xml
PNG5ske_multipercentile_validation.png.gz Display(164.75 KB)
5ske_multipercentile_validation.png
SVG5ske_multipercentile_validation.svg.gz Display(923.00 B)
5ske_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)5ske_validation_2fo-fc_map_coef.cif.gz Display(1.22 MB)
5ske_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)5ske_validation_fo-fc_map_coef.cif.gz Display(1.22 MB)
5ske_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)5ske_validation_2fo-fc_map_coef.mtz Visualize(1.86 MB)
fo-fc (MTZ)5ske_validation_fo-fc_map_coef.mtz Visualize(1.86 MB)

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PDB entries from 2026-01-14

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