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5SK5

CRYSTAL STRUCTURE OF HUMAN PHOSPHODIESTERASE 10 IN COMPLEX WITH C(=O)(N1CCOCC1)c5c(C(Nc3cc2nc(cn2cc3)c4ccccc4)=O)n(nc5)C, micromolar IC50=0.000072

Resources
File formatFile name (file size)
PDBx/mmCIF5sk5.cif.gz Display(278.91 KB)
5sk5.cif
PDBx/mmJSONall5sk5.json.gz Display (Tree)(172.81 KB)
5sk5.json
no-atom5sk5-noatom.json.gz Display (Header)(21.15 KB)
5sk5-noatom.json
add only5sk5-plus.json.gz Display(1.00 KB)
5sk5-plus.json
PDBMLall5sk5.xml.gz Display(382.09 KB)
5sk5.xml
no-atom5sk5-noatom.xml.gz Display(57.01 KB)
5sk5-noatom.xml
ext-atom5sk5-extatom.xml.gz Display(245.93 KB)
5sk5-extatom.xml
pdb_nextgenallpdb_00005sk5_xyz-enrich.cif.gz Display(304.81 KB)
pdb_00005sk5_xyz-enrich.cif
no-atompdb_00005sk5_xyz-no-atom-enrich.xml.gz Display(70.25 KB)
pdb_00005sk5_xyz-no-atom-enrich.xml
ng-only5sk5-plus.json.gz Display(3.41 KB)
5sk5-plus.json
PDBpdb5sk5.ent.gz Display(224.35 KB)
pdb5sk5.ent
RDF5sk5.rdf.gz Visualize(154.20 KB)
5sk5.rdf
Structure factorsr5sk5sf.ent.gz Display(13.09 MB)
r5sk5sf.ent
Biological unit (mmCIF format)5sk5-assembly1.cif.gz Display(72.02 KB)
5sk5-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

5sk5-assembly2.cif.gz Display(72.86 KB)
5sk5-assembly2.cif (B)

*author defined assembly, 1 molecule(s) (monomeric)

5sk5-assembly3.cif.gz Display(71.88 KB)
5sk5-assembly3.cif (C)

*author defined assembly, 1 molecule(s) (monomeric)

5sk5-assembly4.cif.gz Display(70.84 KB)
5sk5-assembly4.cif (D)

*author defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)5sk5.pdb1.gz Display(57.33 KB)
5sk5.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

5sk5.pdb2.gz Display(57.36 KB)
5sk5.pdb2 (B)

*author defined assembly, 1 molecule(s) (monomeric)

5sk5.pdb3.gz Display(57.34 KB)
5sk5.pdb3 (C)

*author defined assembly, 1 molecule(s) (monomeric)

5sk5.pdb4.gz Display(56.50 KB)
5sk5.pdb4 (D)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF5sk5_validation.pdf.gz Display(1.32 MB)
5sk5_validation.pdf
PDF-full5sk5_full_validation.pdf.gz Display(1.33 MB)
5sk5_full_validation.pdf
mmCIF5sk5_validation.cif.gz Display(79.57 KB)
5sk5_validation.cif
XML5sk5_validation.xml.gz Display(60.86 KB)
5sk5_validation.xml
PNG5sk5_multipercentile_validation.png.gz Display(164.71 KB)
5sk5_multipercentile_validation.png
SVG5sk5_multipercentile_validation.svg.gz Display(955.00 B)
5sk5_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)5sk5_validation_2fo-fc_map_coef.cif.gz Display(1.71 MB)
5sk5_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)5sk5_validation_fo-fc_map_coef.cif.gz Display(1.70 MB)
5sk5_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)5sk5_validation_2fo-fc_map_coef.mtz Visualize(2.68 MB)
fo-fc (MTZ)5sk5_validation_fo-fc_map_coef.mtz Visualize(2.68 MB)

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PDB entries from 2026-01-14

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