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5SK1

CRYSTAL STRUCTURE OF HUMAN PHOSPHODIESTERASE 10 IN COMPLEX WITH c12nc(cn1ccc(n2)NC(c3c(C(=O)NC)cnn3C)=O)c4ccccc4, micromolar IC50=0.01331975

Resources
File formatFile name (file size)
PDBx/mmCIF5sk1.cif.gz Display(271.76 KB)
5sk1.cif
PDBx/mmJSONall5sk1.json.gz Display (Tree)(167.65 KB)
5sk1.json
no-atom5sk1-noatom.json.gz Display (Header)(19.89 KB)
5sk1-noatom.json
add only5sk1-plus.json.gz Display(1.00 KB)
5sk1-plus.json
PDBMLall5sk1.xml.gz Display(371.90 KB)
5sk1.xml
no-atom5sk1-noatom.xml.gz Display(54.30 KB)
5sk1-noatom.xml
ext-atom5sk1-extatom.xml.gz Display(240.42 KB)
5sk1-extatom.xml
pdb_nextgenallpdb_00005sk1_xyz-enrich.cif.gz Display(296.89 KB)
pdb_00005sk1_xyz-enrich.cif
no-atompdb_00005sk1_xyz-no-atom-enrich.xml.gz Display(67.43 KB)
pdb_00005sk1_xyz-no-atom-enrich.xml
ng-only5sk1-plus.json.gz Display(3.41 KB)
5sk1-plus.json
PDBpdb5sk1.ent.gz Display(219.65 KB)
pdb5sk1.ent
RDF5sk1.rdf.gz Visualize(148.41 KB)
5sk1.rdf
Structure factorsr5sk1sf.ent.gz Display(9.25 MB)
r5sk1sf.ent
Biological unit (mmCIF format)5sk1-assembly1.cif.gz Display(70.46 KB)
5sk1-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

5sk1-assembly2.cif.gz Display(71.24 KB)
5sk1-assembly2.cif (B)

*author defined assembly, 1 molecule(s) (monomeric)

5sk1-assembly3.cif.gz Display(69.36 KB)
5sk1-assembly3.cif (C)

*author defined assembly, 1 molecule(s) (monomeric)

5sk1-assembly4.cif.gz Display(68.59 KB)
5sk1-assembly4.cif (D)

*author defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)5sk1.pdb1.gz Display(56.35 KB)
5sk1.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

5sk1.pdb2.gz Display(56.44 KB)
5sk1.pdb2 (B)

*author defined assembly, 1 molecule(s) (monomeric)

5sk1.pdb3.gz Display(55.94 KB)
5sk1.pdb3 (C)

*author defined assembly, 1 molecule(s) (monomeric)

5sk1.pdb4.gz Display(55.13 KB)
5sk1.pdb4 (D)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF5sk1_validation.pdf.gz Display(1.31 MB)
5sk1_validation.pdf
PDF-full5sk1_full_validation.pdf.gz Display(1.33 MB)
5sk1_full_validation.pdf
mmCIF5sk1_validation.cif.gz Display(72.59 KB)
5sk1_validation.cif
XML5sk1_validation.xml.gz Display(56.08 KB)
5sk1_validation.xml
PNG5sk1_multipercentile_validation.png.gz Display(169.40 KB)
5sk1_multipercentile_validation.png
SVG5sk1_multipercentile_validation.svg.gz Display(976.00 B)
5sk1_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)5sk1_validation_2fo-fc_map_coef.cif.gz Display(1.03 MB)
5sk1_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)5sk1_validation_fo-fc_map_coef.cif.gz Display(1.01 MB)
5sk1_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)5sk1_validation_2fo-fc_map_coef.mtz Visualize(1.62 MB)
fo-fc (MTZ)5sk1_validation_fo-fc_map_coef.mtz Visualize(1.62 MB)

246905

PDB entries from 2025-12-31

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