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5SK0

CRYSTAL STRUCTURE OF HUMAN PHOSPHODIESTERASE 10 IN COMPLEX WITH N2(c1ccc(cn1)Cl)CC[C@H](C2)NC(c3nn(cc3c4ccncc4)C)=O, micromolar IC50=0.708457

Resources
File formatFile name (file size)
PDBx/mmCIF5sk0.cif.gz Display(280.04 KB)
5sk0.cif
PDBx/mmJSONall5sk0.json.gz Display (Tree)(172.59 KB)
5sk0.json
no-atom5sk0-noatom.json.gz Display (Header)(21.45 KB)
5sk0-noatom.json
add only5sk0-plus.json.gz Display(1015.00 B)
5sk0-plus.json
PDBMLall5sk0.xml.gz Display(381.69 KB)
5sk0.xml
no-atom5sk0-noatom.xml.gz Display(57.41 KB)
5sk0-noatom.xml
ext-atom5sk0-extatom.xml.gz Display(245.64 KB)
5sk0-extatom.xml
pdb_nextgenallpdb_00005sk0_xyz-enrich.cif.gz Display(305.80 KB)
pdb_00005sk0_xyz-enrich.cif
no-atompdb_00005sk0_xyz-no-atom-enrich.xml.gz Display(70.63 KB)
pdb_00005sk0_xyz-no-atom-enrich.xml
ng-only5sk0-plus.json.gz Display(3.42 KB)
5sk0-plus.json
PDBpdb5sk0.ent.gz Display(224.57 KB)
pdb5sk0.ent
RDF5sk0.rdf.gz Visualize(154.09 KB)
5sk0.rdf
Structure factorsr5sk0sf.ent.gz Display(18.04 MB)
r5sk0sf.ent
Biological unit (mmCIF format)5sk0-assembly1.cif.gz Display(72.62 KB)
5sk0-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

5sk0-assembly2.cif.gz Display(72.87 KB)
5sk0-assembly2.cif (B)

*author defined assembly, 1 molecule(s) (monomeric)

5sk0-assembly3.cif.gz Display(73.30 KB)
5sk0-assembly3.cif (C)

*author defined assembly, 1 molecule(s) (monomeric)

5sk0-assembly4.cif.gz Display(70.16 KB)
5sk0-assembly4.cif (D)

*author defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)5sk0.pdb1.gz Display(57.39 KB)
5sk0.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

5sk0.pdb2.gz Display(57.60 KB)
5sk0.pdb2 (B)

*author defined assembly, 1 molecule(s) (monomeric)

5sk0.pdb3.gz Display(57.81 KB)
5sk0.pdb3 (C)

*author defined assembly, 1 molecule(s) (monomeric)

5sk0.pdb4.gz Display(55.45 KB)
5sk0.pdb4 (D)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF5sk0_validation.pdf.gz Display(1.32 MB)
5sk0_validation.pdf
PDF-full5sk0_full_validation.pdf.gz Display(1.34 MB)
5sk0_full_validation.pdf
mmCIF5sk0_validation.cif.gz Display(80.11 KB)
5sk0_validation.cif
XML5sk0_validation.xml.gz Display(60.54 KB)
5sk0_validation.xml
PNG5sk0_multipercentile_validation.png.gz Display(167.11 KB)
5sk0_multipercentile_validation.png
SVG5sk0_multipercentile_validation.svg.gz Display(925.00 B)
5sk0_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)5sk0_validation_2fo-fc_map_coef.cif.gz Display(1.63 MB)
5sk0_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)5sk0_validation_fo-fc_map_coef.cif.gz Display(1.63 MB)
5sk0_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)5sk0_validation_2fo-fc_map_coef.mtz Visualize(2.48 MB)
fo-fc (MTZ)5sk0_validation_fo-fc_map_coef.mtz Visualize(2.48 MB)

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PDB entries from 2026-01-14

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